SCHEMBL5111292

SCHEMBL5111292

O=c1oc2ccccc2c(O)c1-c1cc2c(=O)oc3ccccc3c2o1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.50
MAOB P27338 2/20 0.50
NQO1 P15559 6/20 0.49
MEN1 O00255 4/20 0.49
KMT2A Q03164 4/20 0.49
CYP3A4 P08684 3/20 0.49
ALDH1A1 P00352 2/20 0.49
ABCB11 O95342 1/20 0.49
LMNA P02545 1/20 0.49
TP53 P04637 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP2C9 P11712 1/20 0.49
TSHR P16473 1/20 0.49
MAPK1 P28482 1/20 0.49
CYP2C19 P33261 1/20 0.49
PDE4D Q08499 1/20 0.49
PCSK7 Q16549 1/20 0.49
GPR35 Q9HC97 1/20 0.49
MAPT P10636 3/20 0.47
PKM P14618 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5111826 0.84 NOX4 (0.57) KDM4ENQO1MEN1KMT2AALDH1A1
SCHEMBL5114480 0.82 MAOA (0.40) KDM4EMAOBNQO1MEN1KMT2A
SCHEMBL5120928 0.82 MAOA (0.46) KDM4EMAOBNQO1MEN1KMT2A
SCHEMBL5115329 0.82 MAOB (0.44) KDM4EMAOBNQO1MEN1KMT2A
SCHEMBL5118497 0.81 ESR2 (0.49) KDM4EMAOBMEN1KMT2ACYP3A4
SCHEMBL5114313 0.79 CA12 (0.52) MAOBNQO1GPR35CA12CA9
SCHEMBL5111547 0.79 MAOA (0.59) KDM4EMAOBNQO1MEN1KMT2A
SCHEMBL5112059 0.79 NQO1 (0.55) MAOBNQO1MEN1KMT2ALMNA
SCHEMBL5125176 0.79 MAOB (0.56) KDM4EMAOBNQO1MEN1KMT2A
SCHEMBL5111346 0.79 NQO1 (0.57) KDM4EMAOBNQO1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 16 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7384975-B2 Substituted furochromenes, preparation thereof and their antiinflammatory action GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. (HR) 2008-06-10 US claimed
US-20060148889-A1 Substituted furochromenes, preparation thereof and their antiinflammatory action PLIVA-ISTRAZIVACKI INSTITUT D.O.O. (HR) 2006-07-06 US claimed
EP-1648902-A1 SUBSTITUTED FUROCHROMENES, PREPARATION THEREOF AND THEIR ANTIINFLAMMATORY ACTION PLIVA-ISTRAZIVACKI INSTITUT d.o.o. (HR) 2006-04-26 EP claimed
WO-2005010007-A1 SUBSTITUTED FUROCHROMENES, PREPARATION THEREOF AND THEIR ANTIINFLAMMATORY ACTION PLIVA- ISTRAZIVACKI INSTITUT D.O.O. (HR) 2005-02-03 WO claimed
EP-3606517-B1 COUMARIN DERIVATIVE AS ANTI-ASTHMATIC AGENT, PHARMACEUTICAL COMPOSITION THEREOF AND USE I NOVA MEDICINSKA ISTRAZIVANJA D O O (HR) 2022-05-25 EP disclosed
US-20210113522-A1 COUMARIN DERIVATIVE AS ANTI-ASTHMATIC AGENT, PHARMACEUTICAL COMPOSITION THEREOF, ITS PREPARATION AND USE I-NOVA MEDICINSKA ISTRAZIVANJA D.O.O. (HR) 2021-04-22 US disclosed
EP-3277692-B1 COUMARIN DERIVATIVE AS ANTIVIRAL AGENT, PHARMACEUTICAL COMPOSITION THEREOF, ITS PREPARATION AND USE I NOVA MEDICINSKA ISTRAZIVANJA D O O (HR) 2019-09-11 EP disclosed
US-10266545-B2 Coumarin derivative as antiviral agent, pharmaceutical composition thereof, its preparation and use I-NOVA MEDICINSKA ISTRAZIVANJA D.O.O. (HR) 2019-04-23 US disclosed
US-20180072752-A1 COUMARIN DERIVATIVE AS ANTIVIRAL AGENT, PHARMACEUTICAL COMPOSITION THEREOF, ITS PREPARATION AND USE I-NOVA MEDICINSKA ISTRAZIVANJA D.O.O. (HR) 2018-03-15 US disclosed
US-20180072752-A1 COUMARIN DERIVATIVE AS ANTIVIRAL AGENT, PHARMACEUTICAL COMPOSITION THEREOF, ITS PREPARATION AND USE I-NOVA MEDICINSKA ISTRAZIVANJA D.O.O. (HR) 2018-03-15 US disclosed
US-7384975-B2 Substituted furochromenes, preparation thereof and their antiinflammatory action GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. (HR) 2008-06-10 US disclosed
US-7384975-B2 Substituted furochromenes, preparation thereof and their antiinflammatory action GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. (HR) 2008-06-10 US disclosed
US-7384975-B2 Substituted furochromenes, preparation thereof and their antiinflammatory action GLAXOSMITHKLINE ISTRAZIVACKI CENTAR ZAGREB D.O.O. (HR) 2008-06-10 US disclosed
US-20060148889-A1 Substituted furochromenes, preparation thereof and their antiinflammatory action PLIVA-ISTRAZIVACKI INSTITUT D.O.O. (HR) 2006-07-06 US disclosed
EP-1648902-A1 SUBSTITUTED FUROCHROMENES, PREPARATION THEREOF AND THEIR ANTIINFLAMMATORY ACTION PLIVA-ISTRAZIVACKI INSTITUT d.o.o. (HR) 2006-04-26 EP disclosed
WO-2005010007-A1 SUBSTITUTED FUROCHROMENES, PREPARATION THEREOF AND THEIR ANTIINFLAMMATORY ACTION PLIVA- ISTRAZIVACKI INSTITUT D.O.O. (HR) 2005-02-03 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060148889-A1 Substituted furochromenes, preparation thereof and their antiinflammatory action CYP11B2, CYP11B1, LTC4S KDM4E 3765/4885MAOB 322/4885NQO1 60/4885
US-20180072752-A1 COUMARIN DERIVATIVE AS ANTIVIRAL AGENT, PHARMACEUTICAL COMPOSITION THEREOF, ITS PREPARATION AND USE CYP3A7, MAVS, SARS1 KDM4E 3007/4885MAOB 3312/4885NQO1 609/4885
US-10266545-B2 Coumarin derivative as antiviral agent, pharmaceutical composition thereof, its preparation and use CYP3A7, MAVS, SARS1 KDM4E 3007/4885MAOB 3312/4885NQO1 609/4885
US-20210113522-A1 COUMARIN DERIVATIVE AS ANTI-ASTHMATIC AGENT, PHARMACEUTICAL COMPOSITION THEREOF, ITS PREPARATION AND USE CYP8B1, CYP4B1, CYP3A7 KDM4E 1836/4885MAOB 3043/4885NQO1 824/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.