SCHEMBL5116215

SCHEMBL5116215

CC(C)(O)c1c(N)cccc1Cl

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.48
TSHR P16473 5/20 0.44
NR4A2 P43354 3/20 0.43
PGR P06401 1/20 0.41
CYP3A4 P08684 3/20 0.41
PIK3CA P42336 1/20 0.41
PDK1 Q15118 2/20 0.35
PDK2 Q15119 2/20 0.35
PDK3 Q15120 2/20 0.35
PDK4 Q16654 2/20 0.35
HSD11B1 P28845 1/20 0.35
POLB P06746 1/20 0.34
JAK1 P23458 1/20 0.33
HPGD P15428 2/20 0.32
HSD17B10 Q99714 2/20 0.32
KEAP1 Q14145 1/20 0.32
CD44 P16070 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2A6 P11509 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7753488 0.88 ALDH1A1 (0.48) ALDH1A1TSHRNR4A2PGRCYP3A4
SCHEMBL3787591 0.83 ALDH1A1 (0.52) ALDH1A1TSHRNR4A2PGRCYP3A4
SCHEMBL7764379 0.78 ALDH1A1 (0.47) ALDH1A1TSHRNR4A2PGRCYP3A4
SCHEMBL9265913 0.77 PGR (0.39) ALDH1A1TSHRPGRCYP3A4PDK1
SCHEMBL1772150 0.77 CD44 (0.48) ALDH1A1TSHRPGRCYP3A4PIK3CA
SCHEMBL24730426 0.75 PDK1 (0.35) ALDH1A1TSHRPDK1PDK2PDK3
SCHEMBL31614918 0.75 CYP3A4 (0.36) ALDH1A1TSHRPGRCYP3A4PIK3CA
SCHEMBL8489151 0.75 GAA (0.40) PDK1PDK2PDK3PDK4HSD11B1
SCHEMBL3786889 0.74 TSHR (0.48) ALDH1A1TSHRNR4A2CYP3A4PIK3CA
SCHEMBL30233483 0.74 TSHR (0.48) ALDH1A1TSHRNR4A2CYP3A4PIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160218301-A1 HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING SAME LG CHEM, LTD. (KR) 2016-07-28 US disclosed
US-20160218301-A1 HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING SAME LG CHEM, LTD. (KR) 2016-07-28 US disclosed
WO-2015046986-A1 HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING SAME 주식회사 엘지화학 2015-04-02 WO disclosed
US-7442696-B2 Mineralocorticoid receptor modulator compounds, processes for their preparation, and their uses LIGAND PHARMACEUTICALS, INC. (US) 2008-10-28 US disclosed
US-20070197520-A1 MINERALOCORTICOID RECEPTOR MODULATOR COMPOUNDS, PROCESSES FOR THEIR PREPARATION, AND THEIR USES LIGAND PHARMACEUTICALS INC. 2007-08-23 US disclosed
WO-2006010142-A2 MINERALOCORTICOID RECEPTOR MODULATOR COMPOUNDS, PROCESSES FOR THEIR PREPARATION, AND THEIR USE LIGAND PHARMACEUTICALS, INC. (US) 2006-01-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160218301-A1 HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING ELEMENT USING SAME CRY1, CRY2, NR2E3 ALDH1A1 252/4885TSHR 3480/4885NR4A2 133/4885
US-20070197520-A1 MINERALOCORTICOID RECEPTOR MODULATOR COMPOUNDS, PROCESSES FOR THEIR PREPARATION, AND THEIR USES NR3C2, MC2R, NR3C1 ALDH1A1 3693/4885TSHR 66/4885NR4A2 166/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.