Toluene

Toluene

SCHEMBL512992

Cc1ccccc1.O=S(=O)(O)O.c1ccncc1

nearest known ligand 0.48

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

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

The experimentally established mechanism targets of Toluene. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.48
LMNA P02545 2/20 0.48
ALOX12 P18054 1/20 0.48
ACHE P22303 1/20 0.48
NAPRT Q6XQN6 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.39
TDP1 Q9NUW8 3/20 0.39
PTGS2 P35354 3/20 0.39
ALDH1A1 P00352 3/20 0.39
KMT2A Q03164 3/20 0.39
MEN1 O00255 2/20 0.39
CES2 O00748 1/20 0.39
CES1 P23141 1/20 0.39
KDM4E B2RXH2 2/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
EGFR P00533 1/20 0.38
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Toluene SCHEMBL6514880 1.00 TSHR (0.48) TSHRLMNAALOX12ACHENAPRT
Toluene SCHEMBL27659900 0.94 LMNA (0.46) TSHRLMNAALOX12ACHENAPRT
Toluene SCHEMBL27713635 0.92 TSHR (0.44) TSHRLMNAALOX12ACHENAPRT
Toluene SCHEMBL2178387 0.89 LMNA (0.61) TSHRLMNAALOX12ACHESMN1; SMN2
Toluene SCHEMBL29249545 0.88 SMN1; SMN2 (0.59) TSHRLMNAALOX12ACHENAPRT
Toluene SCHEMBL27551962 0.87 TSHR (0.48) TSHRLMNAALOX12ACHENAPRT
Toluene SCHEMBL22071089 0.87 ALDH1A1 (0.55) TSHRLMNANAPRTSMN1; SMN2TDP1
Toluene SCHEMBL16986055 0.86 PTGS1 (0.37) TSHRLMNAALOX12ACHETDP1
Toluene SCHEMBL248686 0.86 LMNA (0.65) TSHRLMNAALOX12ACHESMN1; SMN2
Toluene SCHEMBL11123126 0.86 LMNA (0.65) TSHRLMNAALOX12ACHESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8367622-B2 Sulfated C-glycoside, method for isolating same and method for synthesizing same SHIZUOKA PREFECTURE PUBLIC UNIVERSITY CORPORATION (JP) 2013-02-05 US disclosed
US-20120029183-A1 SULFATED C-GLYCOSIDE, METHOD FOR ISOLATING SAME AND METHOD FOR SYNTHESIZING SAME SHIZUOKA PREFECTURE PUBLIC UNIVERSITY CORPORATION (JP) 2012-02-02 US disclosed
EP-2385049-A1 SULFATED C-GLYCOSIDE, METHOD FOR ISOLATING SAME AND METHOD FOR SYNTHESIZING SAME Shizuoka Prefecture Public University Corporation (JP) 2011-11-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120029183-A1 SULFATED C-GLYCOSIDE, METHOD FOR ISOLATING SAME AND METHOD FOR SYNTHESIZING SAME ADH1C, ADH1A, CYP21A2 TSHR 1373/4885LMNA 4345/4885ALOX12 2364/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.