SCHEMBL5133149

SCHEMBL5133149

COCCOc1c(C(=O)C(O)c2ccccc2)cccc1S(C)(=O)=O

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCAT2 O15382 1/20 0.39
TSHR P16473 1/20 0.37
LMNA P02545 4/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
HPGD P15428 3/20 0.34
KDM4E B2RXH2 2/20 0.34
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 1/20 0.34
HSD17B10 Q99714 1/20 0.34
MAPK1 P28482 2/20 0.34
PABPC1 P11940 1/20 0.33
EIF4H Q15056 1/20 0.33
KEAP1 Q14145 1/20 0.33
NFE2L2 Q16236 1/20 0.33
ITGB1 P05556 1/20 0.32
ITGA4 P13612 1/20 0.32
KCNA5 P22460 1/20 0.32
AURKA O14965 1/20 0.32
RPS6KB1 P23443 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4430478 0.82 BCAT2 (0.42) BCAT2TSHRHPGDKDM4EALDH1A1
SCHEMBL3631033 0.78 BCAT2 (0.51) BCAT2LMNACES2CES1HPGD
SCHEMBL29384 0.69 USP2 (0.52) LMNACES2CES1HPGDKDM4E
SCHEMBL646150 0.69 PTGER4 (0.35) TSHRALDH1A1MAPK1
Bicarbonate SCHEMBL31648960 0.68 USP2 (0.51) LMNACES2CES1HPGDKDM4E
Bicarbonate SCHEMBL1969232 0.68 USP2 (0.51) LMNACES2CES1HPGDKDM4E
SCHEMBL28827502 0.68 LMNA (0.45) LMNACES2CES1HPGDKDM4E
Methoxymethane SCHEMBL28122245 0.68 USP2 (0.51) LMNACES2CES1HPGDKDM4E
SCHEMBL28102736 0.68 ALDH1A1 (0.46) LMNACES2CES1HPGDKDM4E
SCHEMBL277752 0.68 LMNA (0.52) TSHRLMNACES2CES1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7319099-B2 Such as 1-{3-fluoro-4-[4-(2-isopropoxy-5-methanesulfonyl benzoyl)-piperazin-1-yl]-phenyl}-ethanone for treatment of psychoses, pain, neurodegenerative disfunction in memory and learning, schizophrenia, dementia, attention deficit disorders, or Alzheimer's disease HOFFMANN-LA ROCHE INC. (US) 2008-01-15 US disclosed
US-20050209241-A1 Benzoyl-piperazine derivatives HOFFMANN-LA ROCHE INC. 2005-09-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050209241-A1 Benzoyl-piperazine derivatives SLC1A2, SLC18A2, SLC6A7 BCAT2 225/4885TSHR 4739/4885LMNA 4719/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.