SCHEMBL5141219

SCHEMBL5141219

CCCC(=CC#N)c1nccs1

nearest known ligand 0.40

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.40
PLA2G4A P47712 3/20 0.34
CCNB2 O95067 1/20 0.32
CCNE2 O96020 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
CCNE1 P24864 1/20 0.32
CDK2 P24941 1/20 0.32
CCNB3 Q8WWL7 1/20 0.32
ADORA2A P29274 1/20 0.32
CYP2C19 P33261 1/20 0.32
CES1 P23141 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
FTO Q9C0B1 1/20 0.31
FBP1 P09467 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13369212 0.87 ALDH1A1 (0.42) ALDH1A1PLA2G4ACES1FTOFBP1
SCHEMBL13369309 0.80 ALDH1A1 (0.52) ALDH1A1CYP2C19SMN1; SMN2FTO
SCHEMBL7535989 0.71 FTO (0.45) ALDH1A1SMN1; SMN2FTO
SCHEMBL7192569 0.71 ALDH1A1 (0.42) ALDH1A1FTO
SCHEMBL5141220 0.69 FTO (0.41) ALDH1A1PLA2G4ACCNB2CCNE2CDK1
Bromide SCHEMBL6329679 0.68 PLA2G4A (0.56) ALDH1A1PLA2G4ACCNB2CCNE2CDK1
SCHEMBL16533076 0.66 ALDH1A1 (0.47) ALDH1A1CYP2C19SMN1; SMN2FTO
SCHEMBL19954102 0.65 FTO (0.40) ALDH1A1FTO
SCHEMBL27563650 0.65 ALDH1A1 (0.50) ALDH1A1PLA2G4AADORA2ACES1SMN1; SMN2
SCHEMBL2042556 0.64 ALDH1A1 (0.49) ALDH1A1PLA2G4ACES1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1966202-A1 HETEROARYL SUBSTITUTED PYRROLOÝ2,3-B¨PYRIDINES AND PYRROLOÝ2,3-B¨PYRIMIDINES AS JANUS KINASE INHIBITORS Incyte Corporation (US) 2008-09-10 EP disclosed
WO-2007070514-A1 HETEROARYL SUBSTITUTED PYRROLO[2,3-B]PYRIDINES AND PYRROLO[2,3-B]PYRIMIDINES AS JANUS KINASE INHIBITORS INCYTE CORPORATION (US) 2007-06-21 WO disclosed