SCHEMBL5164020

SCHEMBL5164020

COc1ccccc1S(=O)(=O)Cc1ccccc1-c1ccc(C)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HSD17B10 Q99714 1/20 0.41
HTR7 P34969 3/20 0.41
HTR6 P50406 1/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
DRD3 P35462 1/20 0.41
SCN9A Q15858 1/20 0.40
SYK P43405 1/20 0.40
KDM4E B2RXH2 2/20 0.40
HPGD P15428 2/20 0.40
MAPK1 P28482 2/20 0.40
ALDH1A1 P00352 1/20 0.40
TP53 P04637 1/20 0.40
MAPT P10636 1/20 0.40
POLB P06746 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5165214 0.81 MEN1 (0.48) TSHRCASP1CASP7SMN1; SMN2HSD17B10
SCHEMBL11135262 0.76 POLB (0.45) TSHRHTR7KDM4EHPGDMAPK1
SCHEMBL29038341 0.73 ALOX5AP (0.46) HTR7ALDH1A1MAPTPOLBCYP2C9
SCHEMBL5164016 0.73 NFE2L2 (0.48) HTR6SYKCYP3A4CYP2C9CYP2C19
SCHEMBL5166737 0.72 L3MBTL1 (0.45) SMN1; SMN2HTR6KDM4EHPGDTP53
SCHEMBL4425113 0.72 SYK (0.56) SMN1; SMN2HTR7SYKKDM4EMAPK1
SCHEMBL28835130 0.71 ALDH1A1 (0.50) SMN1; SMN2HTR6KDM4EALDH1A1POLB
SCHEMBL4247206 0.70 HTR6 (0.58) SMN1; SMN2HTR6KDM4ETP53POLB
SCHEMBL13370774 0.70 HTR6 (0.58) SMN1; SMN2HTR6KDM4ETP53GLA
SCHEMBL5165342 0.70 ALDH1A1 (0.52) SMN1; SMN2HSD17B10HTR7HPGDALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1765332-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES Cengent Therapeutics, Inc. (US) 2007-03-28 EP disclosed
WO-2006009876-A2 TRISUBSTITUTED NITROGEN MODULATORS OF TYROSINE PHOSPHATASES CENGENT THERAPEUTICS, INC. (US) 2006-01-26 WO disclosed