SCHEMBL5185609

SCHEMBL5185609

CC(C)n1sc(-c2ccccc2)c(NCCc2cccnc2)c1=O

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
GBA1 P04062 2/20 0.42
F2 P00734 1/20 0.39
KMT2A Q03164 3/20 0.38
MEN1 O00255 2/20 0.38
PDE5A O76074 2/20 0.38
PTAFR P25105 2/20 0.38
HTT P42858 1/20 0.38
TP53 P04637 1/20 0.38
KDM6B O15054 1/20 0.37
KDM4C Q9H3R0 1/20 0.37
JAK2 O60674 1/20 0.37
PTK2 Q05397 1/20 0.37
GSK3B P49841 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5197239 0.88 GSK3B (0.43) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL5184337 0.81 MAOA (0.42) ALDH1A1KMT2AMEN1HTT
SCHEMBL3544822 0.76 TOP2A (0.42) ALDH1A1MAPTSMN1; SMN2KMT2AMEN1
SCHEMBL5224541 0.74 GBA1 (0.44) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2000744 0.70 GBA1 (0.42) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL17844229 0.70 MEN1 (0.48) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL5307781 0.66 LTA4H (0.69) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2733241 0.63 CHRNA7 (0.52)
SCHEMBL12286471 0.62 ACHE (0.52) ALDH1A1NPC1MAPTRAB9ASMN1; SMN2
SCHEMBL2943040 0.62 PIK3CD (0.70) JAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1838687-A1 NON-ANILINIC DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS AstraZeneca AB (SE) 2007-10-03 EP claimed
WO-2006073366-A1 NON-ANILINIC DERIVATIVES OF ISOTHIAZOL-3(2H)-ONE 1,1-DIOXIDES AS LIVER X RECEPTOR MODULATORS ASTRAZENECA AB (SE) 2006-07-13 WO claimed
WO-2016100619-A2 TREATMENT AND DIAGNOSIS OF CANCER RGENIX, INC. (US) 2016-06-23 WO disclosed