SCHEMBL5193832

SCHEMBL5193832

Cc1ccc(CN2CCN(C(=O)c3cccnc3)CC2CC(N)=O)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP6 P51161 1/20 0.46
GAA P10253 1/20 0.44
KDM4E B2RXH2 2/20 0.43
ALDH1A1 P00352 2/20 0.43
POLB P06746 1/20 0.43
PKM P14618 1/20 0.43
MAPK1 P28482 1/20 0.43
CHRM2 P08172 1/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA9 Q16790 2/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
TDP1 Q9NUW8 2/20 0.43
MAPT P10636 2/20 0.42
HTT P42858 1/20 0.42
MYC P01106 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNB4 P30926 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5192328 0.90 TDP1 (0.52) KDM4EALDH1A1POLBMEN1KMT2A
SCHEMBL5206464 0.80 POLB (0.51) KDM4EALDH1A1POLBMAPK1TDP1
SCHEMBL5195325 0.72 SIGMAR1 (0.59) KDM4EALDH1A1POLBPKMMEN1
SCHEMBL5192047 0.72 KMT2A (0.45) FABP6GAAALDH1A1PKMMAPK1
SCHEMBL5191096 0.71 ALDH1A1 (0.46) KDM4EALDH1A1PKMMAPK1
SCHEMBL5193328 0.70 L3MBTL1 (0.49) GAAKDM4EALDH1A1POLBMAPK1
SCHEMBL5190965 0.70 CHRNB2 (0.51) GAAALDH1A1POLBPKMMAPK1
SCHEMBL5199484 0.70 MAPT (0.51) POLBPKMMEN1KMT2AMAPT
SCHEMBL5191582 0.70 TP53 (0.56) POLBPKMMEN1KMT2AMAPT
SCHEMBL5206469 0.70 POLB (0.50) GAAKDM4EALDH1A1POLBTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP claimed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP claimed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO claimed