SCHEMBL5205671

SCHEMBL5205671

C#CCn1cc(C2CCN(C(=O)COc3ccc(Cl)cc3)C2)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 5/20 0.47
ALDH1A1 P00352 5/20 0.47
SMN1; SMN2 Q16637 5/20 0.47
GAA P10253 3/20 0.47
RAB9A P51151 3/20 0.47
L3MBTL1 Q9Y468 2/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
HTT P42858 1/20 0.47
POLB P06746 2/20 0.45
HPGD P15428 1/20 0.45
TP53 P04637 2/20 0.44
HRH2 P25021 1/20 0.44
ATF4 P18848 1/20 0.44
KMT2A Q03164 4/20 0.43
MEN1 O00255 3/20 0.43
GPR183 P32249 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4859500 0.87 KMT2A (0.52) MAPTALDH1A1SMN1; SMN2GAARAB9A
SCHEMBL5205873 0.85 HRH2 (0.51) MAPTALDH1A1SMN1; SMN2GAARAB9A
SCHEMBL5203803 0.79 MAPT (0.52) MAPTALDH1A1SMN1; SMN2GAARAB9A
SCHEMBL5206944 0.74 RAB9A (0.55) MAPTALDH1A1SMN1; SMN2GAARAB9A
SCHEMBL5818040 0.74 SLC2A1 (0.47) MAPTALDH1A1SMN1; SMN2GAARAB9A
SCHEMBL5203557 0.73 ALDH1A1 (0.50) ALDH1A1GAARAB9AL3MBTL1HRH2
SCHEMBL5203814 0.71 SMO (0.51) MAPTALDH1A1CYP3A4HTTPOLB
SCHEMBL5204486 0.70 MAPT (0.54) MAPTALDH1A1SMN1; SMN2RAB9AHTT
SCHEMBL5203232 0.69 LMNA (0.51) MAPTALDH1A1RAB9AHTTPOLB
SCHEMBL5202233 0.69 HRH2 (0.41) MAPTALDH1A1RAB9APOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed