SCHEMBL5203433

SCHEMBL5203433

CCCCn1cc(C2CCN(C(=O)c3cc(C(F)(F)F)ccc3Cl)C2)c2ccccc21

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
TPSAB1 Q15661 5/20 0.50
HRH2 P25021 3/20 0.47
HTR2A P28223 1/20 0.45
HTR2C P28335 1/20 0.45
HTR2B P41595 1/20 0.45
KMT2A Q03164 1/20 0.43
RORC P51449 2/20 0.41
CNR1 P21554 1/20 0.41
CNR2 P34972 1/20 0.41
CRHR1 P34998 3/20 0.41
CRHR2 Q13324 1/20 0.41
PROKR1 Q8TCW9 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5204500 0.92 TPSAB1 (0.47) TPSAB1HRH2KMT2ARORCCNR1
SCHEMBL5203872 0.80 TPSAB1 (0.48) TPSAB1HRH2HTR2AHTR2CHTR2B
SCHEMBL5204533 0.78 ALDH1A1 (0.46) TPSAB1HRH2KMT2APROKR1
SCHEMBL5204952 0.77 HRH2 (0.55) TPSAB1HRH2HTR2AHTR2CHTR2B
SCHEMBL4853030 0.77 HDAC3 (0.46) HRH2HTR2AHTR2CHTR2B
SCHEMBL5204238 0.76 HSD11B1 (0.47) HTR2BKMT2A
SCHEMBL5205803 0.76 HRH2 (0.50) TPSAB1HRH2HTR2AHTR2CHTR2B
SCHEMBL4862667 0.75 TSHR (0.47) TPSAB1HRH2KMT2ACNR2PROKR1
SCHEMBL4862016 0.75 SLC5A1 (0.49)
SCHEMBL4859740 0.75 HTR2A (0.46) TPSAB1HRH2HTR2AHTR2CHTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed