Trifluoroacetic Acid

Trifluoroacetic Acid

SCHEMBL5205467

N#Cc1ccc(CN(C(=O)CCC(=O)NCc2ccccn2)c2ccccc2Oc2cccc(CN)c2)cc1.O=C(O)C(F)(F)F

nearest known ligand 0.39

Full drug profile on Sugi Atlas →

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.39
KMT2A Q03164 2/20 0.38
CACNA1B Q00975 2/20 0.37
HPGD P15428 1/20 0.37
ALOX15 P16050 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
ALDH1A1 P00352 1/20 0.37
LOX P28300 2/20 0.36
LOXL2 Q9Y4K0 2/20 0.36
MEN1 O00255 1/20 0.35
MAPK1 P28482 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Trifluoroacetic Acid SCHEMBL5201682 0.92 ALDH1A1 (0.40) KMT2ACACNA1BHPGDALOX15TDP1
Trifluoroacetic Acid SCHEMBL5202243 0.89 EPHX2 (0.36) CACNA1BTDP1ALDH1A1LOXLOXL2
Trifluoroacetic Acid SCHEMBL5201746 0.88 CACNA1B (0.36) KMT2ACACNA1BALDH1A1LOXLOXL2
Trifluoroacetic Acid SCHEMBL5208477 0.88 ALDH1A1 (0.37) KMT2ACACNA1BALDH1A1LOXLOXL2
Trifluoroacetic Acid SCHEMBL5202153 0.88 TSPO (0.41) SCN9AKMT2AHPGDALDH1A1MEN1
Trifluoroacetic Acid SCHEMBL5204751 0.88 TPSAB1 (0.35) KMT2ACACNA1BTDP1ALDH1A1LOX
Trifluoroacetic Acid SCHEMBL5207958 0.87 SMN1; SMN2 (0.47) KMT2AHPGDTDP1ALDH1A1MEN1
Trifluoroacetic Acid SCHEMBL5208348 0.87 RAB9A (0.37) SCN9AKMT2ACACNA1BLOXLOXL2
Trifluoroacetic Acid SCHEMBL5207856 0.86 KMT2A (0.37) KMT2AHPGDALOX15TDP1ALDH1A1
Trifluoroacetic Acid SCHEMBL5207332 0.85 TPSAB1 (0.44) KMT2AALDH1A1LOXLOXL2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7160887-B1 Aromatic amine derivatives, their production and use TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-09 US disclosed
EP-1123918-B1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME TAKEDA PHARMACEUTICAL (JP) 2005-03-09 EP disclosed
EP-1123918-A1 AROMATIC AMINE DERIVATIVES, PROCESS FOR THE PREPARATION THEREOF AND AGENTS CONTAINING THE SAME Takeda Chemical Industries, Ltd. (JP) 2001-08-16 EP disclosed