SCHEMBL5205864

SCHEMBL5205864

Cn1cc(C2CCN(C(=O)c3cccnc3)C2)c2ccccc21

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RORC P51449 1/20 0.46
GAA P10253 1/20 0.46
ALDH1A1 P00352 6/20 0.46
HTT P42858 2/20 0.46
KDM4E B2RXH2 1/20 0.46
CCR5 P51681 1/20 0.46
HSD11B1 P28845 2/20 0.45
USP2 O75604 1/20 0.45
SPR P35270 1/20 0.44
HPGDS O60760 1/20 0.44
CHRNB2 P17787 1/20 0.44
CHRNB4 P30926 1/20 0.44
CHRNA3 P32297 1/20 0.44
CHRNA7 P36544 1/20 0.44
CHRNA4 P43681 1/20 0.44
PDE2A O00408 1/20 0.44
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.43
AXL P30530 1/20 0.43
FLT3 P36888 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5203268 0.87 GAA (0.48) GAAALDH1A1HTTKDM4ECCR5
SCHEMBL5201722 0.82 HTR2B (0.53) RORCALDH1A1USP2HPGDMAPK1
SCHEMBL4859672 0.80 HSD11B1 (0.52) HSD11B1SPRDRD2DRD3
SCHEMBL5203887 0.79 ALDH1A1 (0.52) GAAALDH1A1KDM4EHSD11B1SPR
SCHEMBL5202338 0.78 GFER (0.47) RORCALDH1A1HSD11B1USP2SPR
SCHEMBL3065644 0.76 HSD11B1 (0.68) ALDH1A1HTTKDM4EHSD11B1HPGDS
SCHEMBL5937364 0.75 ALDH1A1 (0.57) RORCALDH1A1KDM4EUSP2SPR
SCHEMBL5705162 0.75 RORC (0.51) RORCALDH1A1KDM4EUSP2SPR
SCHEMBL14730730 0.73 RECQL (0.59) GAAALDH1A1HTTCHRNB2CHRNB4
SCHEMBL14197788 0.73 RECQL (0.59) GAAALDH1A1HTTCHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed