SCHEMBL5203887

SCHEMBL5203887

CSc1ncccc1C(=O)N1CCC(c2cn(C)c3ccccc23)C1

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.52
KMT2A Q03164 3/20 0.52
HSD11B1 P28845 2/20 0.52
LMNA P02545 2/20 0.51
MEN1 O00255 2/20 0.51
KDM4E B2RXH2 1/20 0.51
GAA P10253 1/20 0.47
SPR P35270 1/20 0.44
TPSAB1 Q15661 1/20 0.43
GFER P55789 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
RAB9A P51151 1/20 0.42
PROKR1 Q8TCW9 1/20 0.41
HCRTR1 O43613 1/20 0.41
POLB P06746 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4859672 0.87 HSD11B1 (0.52) HSD11B1SPRTPSAB1GFERPROKR1
SCHEMBL5203557 0.85 ALDH1A1 (0.50) ALDH1A1KMT2AHSD11B1LMNAMEN1
SCHEMBL5205864 0.79 RORC (0.46) ALDH1A1KMT2AHSD11B1MEN1KDM4E
SCHEMBL5201936 0.79 SPR (0.39) ALDH1A1KMT2AHSD11B1LMNAMEN1
SCHEMBL5202338 0.76 GFER (0.47) ALDH1A1HSD11B1SPRTPSAB1GFER
SCHEMBL5201722 0.75 HTR2B (0.53) ALDH1A1KMT2ALMNAMEN1RAB9A
SCHEMBL5937364 0.72 ALDH1A1 (0.57) ALDH1A1KMT2ALMNAKDM4ESPR
SCHEMBL5705162 0.72 RORC (0.51) ALDH1A1KMT2ALMNAMEN1KDM4E
SCHEMBL29944450 0.72 KMT2A (0.73) ALDH1A1KMT2ALMNAMEN1KDM4E
SCHEMBL4858050 0.70 RAB9A (0.62) ALDH1A1KMT2ALMNAMEN1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed