SCHEMBL5206008

SCHEMBL5206008

Cc1cc(C)cc(Cn2cc(C3CCN(CC(=O)Nc4scc(C)c4C#N)C3)c3ccccc32)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH2 P25021 6/20 0.41
DRD4 P21917 3/20 0.40
HTR2A P28223 4/20 0.38
HTR2C P28335 4/20 0.38
HTR2B P41595 4/20 0.38
HTR6 P50406 2/20 0.38
SMO Q99835 1/20 0.37
DRD2 P14416 1/20 0.37
HDAC3 O15379 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC2 Q92769 1/20 0.36
HDAC10 Q969S8 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
HDAC6 Q9UBN7 1/20 0.36
NCOR2 Q9Y618 1/20 0.36
POLB P06746 1/20 0.36
MAPT P10636 1/20 0.36
RAC1 P63000 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
TP53 P04637 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4857534 0.89 DRD4 (0.40) HRH2DRD4POLBMAPTSMN1; SMN2
SCHEMBL5203876 0.68 ALDH1A1 (0.39) HRH2DRD4HTR2AHTR2CHTR2B
SCHEMBL4859877 0.67 HRH2 (0.42) HRH2HTR2AHTR2CHTR2BHTR6
SCHEMBL4859724 0.63 SMO (0.46) HRH2HTR2AHTR2CHTR2BHTR6
SCHEMBL5203814 0.62 SMO (0.51) HRH2HTR2AHTR2CHTR2BHTR6
SCHEMBL5347587 0.62 CYP1A2 (0.50) HRH2HTR2AHTR2CHTR2BHTR6
SCHEMBL5202142 0.61 LMNA (0.50) HRH2HTR6SMODRD2HDAC3
SCHEMBL5205062 0.61 SMO (0.46) HRH2SMOHDAC3HDAC1HDAC2
SCHEMBL5202270 0.61 MAPT (0.43) DRD4MAPTSMN1; SMN2TP53MEN1
SCHEMBL5350498 0.61 HRH2 (0.76) HRH2HTR2AHTR2CHTR2BHTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed