SCHEMBL5206419

SCHEMBL5206419

CCn1cc(C2CCN(C(=O)c3ccc(F)cc3F)C2)c2ccccc21

nearest known ligand 0.49

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 2/20 0.49
ALDH1A1 P00352 1/20 0.49
HSD11B1 P28845 2/20 0.48
TPSAB1 Q15661 2/20 0.47
UBE2M P61081 1/20 0.46
DCUN1D1 Q96GG9 1/20 0.46
SLC2A1 P11166 1/20 0.45
KMT2A Q03164 2/20 0.45
HRH2 P25021 2/20 0.44
CNR1 P21554 2/20 0.43
RBP4 P02753 1/20 0.43
PROKR1 Q8TCW9 1/20 0.43
DPP4 P27487 1/20 0.43
MAPK1 P28482 1/20 0.42
HTR2A P28223 1/20 0.42
HTR2C P28335 1/20 0.42
GFER P55789 1/20 0.42
MEN1 O00255 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4860093 0.88 ALDH1A1 (0.45) SMN1; SMN2ALDH1A1HSD11B1TPSAB1SLC2A1
SCHEMBL5203757 0.86 NPC1 (0.57) SMN1; SMN2ALDH1A1HSD11B1TPSAB1SLC2A1
SCHEMBL5202510 0.83 HSD11B1 (0.55) SMN1; SMN2ALDH1A1HSD11B1TPSAB1KMT2A
SCHEMBL5202100 0.80 ALDH1A1 (0.51) SMN1; SMN2ALDH1A1HSD11B1TPSAB1KMT2A
SCHEMBL5202168 0.80 PROKR1 (0.47) SMN1; SMN2ALDH1A1TPSAB1SLC2A1KMT2A
SCHEMBL5204500 0.80 TPSAB1 (0.47) SMN1; SMN2ALDH1A1TPSAB1KMT2AHRH2
SCHEMBL4859715 0.79 HCRTR1 (0.41) SMN1; SMN2ALDH1A1TPSAB1SLC2A1KMT2A
SCHEMBL5204533 0.78 ALDH1A1 (0.46) SMN1; SMN2ALDH1A1HSD11B1TPSAB1KMT2A
SCHEMBL4854486 0.78 ALDH1A1 (0.46) ALDH1A1HSD11B1KMT2AHRH2MEN1
SCHEMBL4862667 0.78 TSHR (0.47) SMN1; SMN2ALDH1A1HSD11B1TPSAB1UBE2M

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP claimed
EP-1654253-B1 SUBSTITUTED 3-PYRROLIDIN-INDOLE DERIVATIVES GRUENENTHAL GMBH (DE) 2007-01-03 EP disclosed