SCHEMBL5195403

SCHEMBL5195403

CN1CCNC(CC(=O)NCc2ccc3c(c2)CCC3)C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
ALOX12 P18054 1/20 0.42
TRPV1 Q8NER1 8/20 0.41
NOS2 P35228 1/20 0.40
MAPK14 Q16539 1/20 0.40
ERCC1 P07992 1/20 0.39
ERCC4 Q92889 1/20 0.39
PPID Q08752 1/20 0.38
HTT P42858 1/20 0.38
NPC1 O15118 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C19 P33261 1/20 0.37
RAB9A P51151 1/20 0.37
NAMPT P43490 1/20 0.37
TP53 P04637 1/20 0.36
ALOX15 P16050 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5214027 0.81 NPC1 (0.53) HPGDNPC1RAB9AMEN1KMT2A
SCHEMBL5208438 0.81 FAAH (0.54) SMN1; SMN2MAPK14NPC1RAB9ANAMPT
SCHEMBL5193934 0.72 ALDH1A1 (0.53) HPGDHTTALOX15MEN1KMT2A
SCHEMBL16250732 0.69 MAPK14 (0.54) HPGDSMN1; SMN2ALOX12MAPK14HTT
SCHEMBL2917177 0.69 REN (0.35) CYP1A2CYP2C19ALOX15LMNA
SCHEMBL5192010 0.68 HPGD (0.46) HPGDSMN1; SMN2NOS2MEN1KMT2A
SCHEMBL27393194 0.68 MAPK14 (0.52) HPGDSMN1; SMN2ALOX12MAPK14HTT
SCHEMBL5191071 0.67 LMNA (0.47) MEN1KMT2ALMNA
SCHEMBL5192873 0.67 LMNA (0.47) MEN1KMT2ALMNA
SCHEMBL20051408 0.67 MAPK14 (0.54) HPGDSMN1; SMN2ALOX12MAPK14HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968206-B8 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX INC (US) 2007-01-24 EP disclosed
EP-0968206-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 2000-01-05 EP disclosed
WO-1998037079-A1 N-HETEROCYCLIC DERIVATIVES AS NOS INHIBITORS BERLEX LABORATORIES, INC. (US) 1998-08-27 WO disclosed