SCHEMBL5219253

SCHEMBL5219253

COc1ccc([N+](=O)[O-])c(N2CCC(NC(=O)O)CC2)n1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TXNRD1 Q16881 6/20 0.47
OPRK1 P41145 2/20 0.45
ALDH1A1 P00352 7/20 0.45
CRHBP P24387 2/20 0.42
CRHR2 Q13324 2/20 0.42
MAPT P10636 4/20 0.41
MAPK1 P28482 2/20 0.41
POLB P06746 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
LMNA P02545 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2689490 0.85 TDP1 (0.52) TXNRD1ALDH1A1MAPTMAPK1POLB
SCHEMBL5752950 0.85 TXNRD1 (0.48) TXNRD1OPRK1ALDH1A1
SCHEMBL3281560 0.82 OPRK1 (0.40) TXNRD1OPRK1ALDH1A1CRHBPCRHR2
Hydrochloric Acid SCHEMBL5220902 0.80 TXNRD1 (0.49) TXNRD1ALDH1A1MAPTMAPK1POLB
SCHEMBL19691739 0.80 TXNRD1 (0.46) TXNRD1ALDH1A1MAPTMAPK1LMNA
SCHEMBL19691737 0.80 TXNRD1 (0.46) TXNRD1ALDH1A1MAPTMAPK1LMNA
SCHEMBL5752857 0.79 ALDH1A1 (0.64) TXNRD1ALDH1A1MAPTMAPK1POLB
SCHEMBL2421463 0.79 ALDH1A1 (0.64) TXNRD1ALDH1A1MAPTMAPK1POLB
SCHEMBL6509373 0.78 TXNRD1 (0.47) TXNRD1ALDH1A1MAPTMAPK1POLB
SCHEMBL30435070 0.77 SIRT6 (0.54) TXNRD1ALDH1A1MAPTMAPK1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1664025-B1 PYRROL DERIVATIVES WITH ANTIBACTERIAL ACTIVITY ASTRAZENECA AB (SE) 2007-09-19 EP disclosed