SCHEMBL5224207

SCHEMBL5224207

CC1CCCN1Cc1cnn(-c2ccc(-c3cccc(F)c3)cc2)c1-c1ccco1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.36
HRH3 Q9Y5N1 6/20 0.35
HTR3A P46098 3/20 0.35
ADRB2 P07550 2/20 0.34
POLB P06746 1/20 0.34
BMPR1B O00238 1/20 0.34
BMPR1A P36894 1/20 0.34
TGFBR1 P36897 1/20 0.34
ACVRL1 P37023 1/20 0.34
ACVR1 Q04771 1/20 0.34
GRM2 Q14416 1/20 0.34
CHRNB1 P11230 1/20 0.34
CHRNB2 P17787 1/20 0.34
CHRNB4 P30926 1/20 0.34
CHRNA3 P32297 1/20 0.34
CHRNB3 Q05901 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5225463 0.86 ALDH1A1 (0.41) HRH3POLB
SCHEMBL5228473 0.85 ALDH1A1 (0.41) HRH3POLBCHRNB1CHRNB2CHRNB4
SCHEMBL5229287 0.82 EGFR (0.40) DHODH
SCHEMBL5224673 0.82 SMO (0.40) DHODH
SCHEMBL5226613 0.82 SMO (0.40) DHODHPOLB
SCHEMBL5226986 0.82 DRD4 (0.39) POLB
SCHEMBL5228047 0.81 HTR2C (0.37) DHODHADRB2
SCHEMBL5224744 0.80 HTR1A (0.38) DHODHHTR3AACVR1
SCHEMBL5227271 0.79 DHODH (0.39) DHODH
SCHEMBL5225471 0.78 HRH3 (0.35) HRH3POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed