SCHEMBL5224696

SCHEMBL5224696

CN(C)CCN(C)Cc1cnn(-c2ccc(-c3ccc(F)cc3)cc2)c1-c1cccc(Cl)c1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.39
NR3C1 P04150 5/20 0.38
NPC1 O15118 2/20 0.37
RAB9A P51151 2/20 0.37
MEN1 O00255 1/20 0.37
PKM P14618 1/20 0.37
KMT2A Q03164 1/20 0.37
TP53 P04637 1/20 0.36
MAPT P10636 1/20 0.36
KCNH2 Q12809 1/20 0.35
PGR P06401 1/20 0.35
LMNA P02545 2/20 0.35
CCR1 P32246 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5232217 0.85 NR3C1 (0.40) TAAR1NR3C1NPC1RAB9ATP53
SCHEMBL5227418 0.79 PTGS1 (0.38) NR3C1NPC1RAB9ATP53MAPT
SCHEMBL5230174 0.78 DRD4 (0.46) PKMTP53MAPT
SCHEMBL5227445 0.78 DRD4 (0.46) NR3C1MAPT
SCHEMBL7257428 0.77 ADORA2A (0.40) NR3C1NPC1RAB9AKMT2ALMNA
SCHEMBL5226500 0.73 PTGS1 (0.36) NR3C1NPC1RAB9ATP53MAPT
SCHEMBL5230607 0.73 DRD4 (0.46) NR3C1TP53MAPT
SCHEMBL5227774 0.73 DRD3 (0.45) TP53MAPT
SCHEMBL5228024 0.71 HTR2C (0.42) NR3C1TP53PGRLMNA
SCHEMBL5228140 0.71 NR3C1 (0.48) NR3C1RAB9AKMT2ATP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed