SCHEMBL5230607

SCHEMBL5230607

Fc1ccc(-c2ccc(-n3ncc(CN4CCN(CCN5CCCC5)CC4)c3-c3cccc(Cl)c3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD4 P21917 5/20 0.46
DRD3 P35462 5/20 0.46
DRD2 P14416 3/20 0.46
SMO Q99835 1/20 0.43
MAPT P10636 3/20 0.40
TP53 P04637 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MCHR1 Q99705 1/20 0.38
FNTA P49354 1/20 0.38
PGGT1B P53609 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CNR1 P21554 1/20 0.38
CNR2 P34972 1/20 0.38
MAPK14 Q16539 1/20 0.37
NR3C1 P04150 1/20 0.37
MAP3K9 P80192 1/20 0.37
MAP3K11 Q16584 1/20 0.37
SLC6A2 P23975 1/20 0.37
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227774 0.99 DRD3 (0.45) DRD4DRD3DRD2SMOMAPT
SCHEMBL5230174 0.91 DRD4 (0.46) DRD4DRD3DRD2SMOMAPT
SCHEMBL5227445 0.89 DRD4 (0.46) DRD4DRD3DRD2SMOMAPT
SCHEMBL5229642 0.88 DRD2 (0.42) DRD4DRD3DRD2SMOMAPT
SCHEMBL5226907 0.87 DRD4 (0.43) DRD4DRD3DRD2SMOMAPT
SCHEMBL5228024 0.82 HTR2C (0.42) DRD4DRD3DRD2SMOTP53
SCHEMBL5223970 0.79 ADORA2A (0.40) DRD4DRD3DRD2SMOMAPT
SCHEMBL5225265 0.78 SMO (0.59) DRD4DRD3DRD2SMOMAPT
SCHEMBL5226797 0.78 SMO (0.61) SMOMAPTALDH1A1L3MBTL1MAPK14
SCHEMBL5229662 0.77 SMO (0.58) DRD4SMOMAPTALDH1A1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed