SCHEMBL5227774

SCHEMBL5227774

Fc1ccc(-c2ccc(-n3ncc(CN4CCN(CCN5CCCCC5)CC4)c3-c3cccc(Cl)c3)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 5/20 0.45
DRD4 P21917 4/20 0.45
DRD2 P14416 3/20 0.45
SMO Q99835 1/20 0.43
MAPT P10636 3/20 0.40
TP53 P04637 1/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
ALDH1A1 P00352 2/20 0.39
MAPK14 Q16539 2/20 0.39
CYP2D6 P10635 1/20 0.38
CYP2C19 P33261 1/20 0.38
MCHR1 Q99705 1/20 0.38
FNTA P49354 1/20 0.38
PGGT1B P53609 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5230607 0.99 DRD4 (0.46) DRD3DRD4DRD2SMOMAPT
SCHEMBL5230174 0.90 DRD4 (0.46) DRD3DRD4DRD2SMOMAPT
SCHEMBL5227445 0.88 DRD4 (0.46) DRD3DRD4DRD2SMOMAPT
SCHEMBL5229642 0.87 DRD2 (0.42) DRD3DRD4DRD2SMOMAPT
SCHEMBL5226907 0.86 DRD4 (0.43) DRD3DRD4DRD2SMOMAPT
SCHEMBL5228024 0.81 HTR2C (0.42) DRD3DRD4DRD2SMOTP53
SCHEMBL5223970 0.78 ADORA2A (0.40) DRD3DRD4DRD2SMOMAPT
SCHEMBL5225265 0.77 SMO (0.59) DRD3DRD4DRD2SMOMAPT
SCHEMBL5226797 0.77 SMO (0.61) SMOMAPTALDH1A1MAPK14CYP2D6
SCHEMBL5229662 0.77 SMO (0.58) DRD4SMOMAPTALDH1A1MAPK14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed