SCHEMBL5228024

SCHEMBL5228024

OC1CCN(Cc2cnn(-c3ccc(-c4ccc(F)cc4)cc3)c2-c2cccc(Cl)c2)C1

nearest known ligand 0.42

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 3/20 0.42
MCHR1 Q99705 3/20 0.42
DRD2 P14416 1/20 0.40
DRD4 P21917 1/20 0.40
DRD3 P35462 1/20 0.40
LMNA P02545 1/20 0.40
TP53 P04637 2/20 0.40
ALPI P09923 1/20 0.39
ALPG P10696 1/20 0.39
SMO Q99835 1/20 0.38
NR3C1 P04150 3/20 0.38
ROCK2 O75116 2/20 0.38
PDE2A O00408 2/20 0.37
PGR P06401 1/20 0.37
USP7 Q93009 1/20 0.37
PDCD1LG2 Q9BQ51 2/20 0.36
CD274 Q9NZQ7 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5227214 0.86 SMO (0.52) LMNASMONR3C1ROCK2
SCHEMBL5227619 0.84 F10 (0.42) HTR2CMCHR1USP7
SCHEMBL5230174 0.83 DRD4 (0.46) DRD2DRD4DRD3TP53ALPI
SCHEMBL5227445 0.83 DRD4 (0.46) DRD2DRD4DRD3SMONR3C1
SCHEMBL5226907 0.83 DRD4 (0.43) MCHR1DRD2DRD4DRD3TP53
SCHEMBL5230607 0.82 DRD4 (0.46) MCHR1DRD2DRD4DRD3TP53
SCHEMBL5224144 0.81 HTR2C (0.38) HTR2CMCHR1SMONR3C1ROCK2
SCHEMBL5227774 0.81 DRD3 (0.45) MCHR1DRD2DRD4DRD3TP53
SCHEMBL2001554 0.79 SMO (0.50) HTR2CMCHR1DRD2DRD4DRD3
SCHEMBL5907351 0.79 F10 (0.44) CD274

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed