SCHEMBL5224860

SCHEMBL5224860

CCN(CC)Cc1cnn(-c2ccc(C3=C(Cc4ccccc4)OCO3)cc2)c1-c1ccco1

nearest known ligand 0.31

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.31
HPGD P15428 3/20 0.31
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 2/20 0.31
MAPT P10636 1/20 0.31
LMNA P02545 2/20 0.31
TSHR P16473 2/20 0.31
ALOX15 P16050 1/20 0.31
MAPK1 P28482 1/20 0.31
HTT P42858 1/20 0.31
PPARD Q03181 1/20 0.30
PPARA Q07869 1/20 0.30
RORC P51449 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5229304 0.91 ALDH1A1 (0.33) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL5226173 0.86 SMO (0.38) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL5222928 0.83 SMO (0.38) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL5226844 0.81 SIGMAR1 (0.34) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL5225471 0.80 HRH3 (0.35) KDM4EPPARDPPARA
SCHEMBL5224853 0.79 HSD17B10 (0.43) ALDH1A1HPGDKDM4EHSD17B10LMNA
SCHEMBL5226667 0.78 DRD4 (0.39) ALDH1A1KDM4ETSHR
SCHEMBL5230408 0.77 SLC2A1 (0.32) ALDH1A1HPGDHSD17B10MAPTLMNA
SCHEMBL5224717 0.77 NPBWR1 (0.45) ALDH1A1HPGDKDM4EHSD17B10MAPT
SCHEMBL5224947 0.76 ALDH1A1 (0.38) ALDH1A1HPGDKDM4EHSD17B10MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed