SCHEMBL5228536

SCHEMBL5228536

O=C1CN(Cc2cnn(-c3ccc(-c4cccc(F)c4)cc3)c2-c2ccco2)CCN1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 2/20 0.38
ERBB2 P04626 2/20 0.38
DHODH Q02127 1/20 0.36
SCN9A Q15858 3/20 0.34
NPSR1 Q6W5P4 1/20 0.34
HTR6 P50406 1/20 0.34
KDM4E B2RXH2 2/20 0.34
SLC2A1 P11166 1/20 0.34
POLB P06746 1/20 0.34
PDCD1 Q15116 1/20 0.34
CD274 Q9NZQ7 1/20 0.34
GRM2 Q14416 1/20 0.34
TP53 P04637 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
MCHR1 Q99705 1/20 0.33
ALDH1A1 P00352 2/20 0.33
USP2 O75604 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5224744 0.90 HTR1A (0.38) EGFRERBB2DHODHHTR6KDM4E
SCHEMBL5230401 0.87 ALDH1A1 (0.38) NPSR1KDM4ESLC2A1POLBPDCD1
SCHEMBL5226613 0.83 SMO (0.40) DHODHKDM4EPOLBTP53SMN1; SMN2
SCHEMBL5224673 0.83 SMO (0.40) DHODHHTR6KDM4EALDH1A1
SCHEMBL5229287 0.81 EGFR (0.40) EGFRERBB2DHODHKDM4EMEN1
SCHEMBL5228047 0.80 HTR2C (0.37) DHODHKDM4EMCHR1ALDH1A1ROCK2
SCHEMBL5226986 0.79 DRD4 (0.39) KDM4EPOLBTP53MCHR1ALDH1A1
SCHEMBL5230408 0.79 SLC2A1 (0.32) EGFRERBB2NPSR1SLC2A1PDCD1
SCHEMBL5226151 0.76 SMO (0.35) KDM4ETP53MEN1KMT2AALDH1A1
SCHEMBL5227271 0.76 DHODH (0.39) DHODHKDM4ETP53SMN1; SMN2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1611122-B1 SUBSTITUTED PYRAZOLE COMPOUNDS MERCK PATENT GMBH (DE) 2007-06-13 EP disclosed