SCHEMBL5230475

SCHEMBL5230475

CNC1(C(C)=O)CN(c2ccncc2)CCN1C(=O)O

nearest known ligand 0.44

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 5/20 0.44
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
CYP3A4 P08684 5/20 0.43
TSHR P16473 2/20 0.42
CYP2C19 P33261 3/20 0.41
HIF1A Q16665 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP2D6 P10635 2/20 0.40
ITGB3 P05106 7/20 0.40
ITGA2B P08514 7/20 0.40
HSD17B10 Q99714 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5238186 0.88 CYP2C19 (0.43) CYP2C9MEN1KMT2ACYP3A4TSHR
SCHEMBL5239779 0.86 MAPT (0.40) CYP2C9MEN1KMT2ACYP2C19ALDH1A1
SCHEMBL5239092 0.85 MEN1 (0.41) MEN1KMT2AALDH1A1
SCHEMBL5232288 0.85 MAPT (0.41) MEN1KMT2AALDH1A1
SCHEMBL5237326 0.84 CA2 (0.43) MEN1KMT2ATSHR
SCHEMBL5236546 0.84 USP2 (0.46) CYP2C9MEN1KMT2ACYP3A4TSHR
SCHEMBL5233064 0.82 L3MBTL1 (0.48) MEN1KMT2AALDH1A1
SCHEMBL5234836 0.81 MEN1 (0.43) CYP2C9MEN1KMT2ACYP3A4CYP2C19
SCHEMBL5235440 0.81 ALDH1A1 (0.40) CYP2C9MEN1KMT2ACYP3A4CYP2C19
SCHEMBL5232372 0.81 ALDH1A1 (0.41) CYP2C9MEN1KMT2ACYP3A4TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1701946-B1 DERIVATIVES OF 1-PIPERAZINE- AND 1-HOMOPIPERAZINE-CARBOXYLATES, PREPARATION METHOD THEREOF AND USE OF SAME AS INHIBITORS OF THE FAAH ENZYME SANOFI AVENTIS (FR) 2007-12-19 EP claimed