SCHEMBL5233398

SCHEMBL5233398

NC(=O)C[C@@H](c1ccccc1)N1CC2CN(C(=O)C3CCN(c4ncccn4)CC3)CC2C1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.44
CYP2C19 P33261 1/20 0.44
RIPK1 Q13546 2/20 0.43
LMNA P02545 4/20 0.43
MAPK1 P28482 3/20 0.43
ALDH1A1 P00352 3/20 0.43
HPGD P15428 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
TSHR P16473 2/20 0.41
HSD17B10 Q99714 2/20 0.41
USP2 O75604 1/20 0.41
TP53 P04637 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
HTT P42858 2/20 0.39
RXFP1 Q9HBX9 1/20 0.39
HTR1A P08908 1/20 0.39
POLB P06746 1/20 0.39
GAA P10253 1/20 0.39
CCL5 P13501 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4689575 0.79 CCR5 (0.47) KDM4ECYP2C19RIPK1LMNAMAPK1
SCHEMBL5229817 0.78 CCR5 (0.42) RIPK1ALDH1A1TDP1CCR5CNR1
SCHEMBL5235073 0.77 CHRNB2 (0.53) RIPK1ALDH1A1SMN1; SMN2L3MBTL1GAA
Cyclopentane SCHEMBL4694323 0.74 CCR5 (0.54) CCL5CCR5
SCHEMBL5234052 0.73 PKM (0.46) KDM4ECYP2C19MAPK1ALDH1A1HPGD
SCHEMBL5235643 0.73 CHRNB2 (0.53) KDM4ECYP2C19LMNAMAPK1ALDH1A1
SCHEMBL5235854 0.73 PARP1 (0.37) CYP2C19MAPK1HPGDTDP1
SCHEMBL5237872 0.73 CCL5 (0.40) CYP2C19LMNAMAPK1ALDH1A1HPGD
SCHEMBL5234640 0.72 HCRTR1 (0.52) MAPK1ALDH1A1
SCHEMBL5233454 0.72 DPP4 (0.49) ALDH1A1HPGDHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed