SCHEMBL5229817

SCHEMBL5229817

NC(=O)C[C@@H](c1ccccc1)N1CC2CN(C(=O)C3CCOC3)CC2C1

nearest known ligand 0.42

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 3/20 0.42
RIPK1 Q13546 1/20 0.39
TDP1 Q9NUW8 1/20 0.37
KCNH2 Q12809 1/20 0.37
NPY5R Q15761 1/20 0.37
ALDH1A1 P00352 1/20 0.37
NAMPT P43490 5/20 0.36
GRM5 P41594 2/20 0.36
CNR1 P21554 1/20 0.35
CNR2 P34972 1/20 0.35
KDM1A O60341 3/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5234052 0.81 PKM (0.46) TDP1ALDH1A1
SCHEMBL5233398 0.78 KDM4E (0.44) CCR5RIPK1TDP1ALDH1A1CNR1
SCHEMBL4691437 0.77 CCR5 (0.54) CCR5RIPK1
SCHEMBL5235854 0.77 PARP1 (0.37) TDP1
SCHEMBL5237872 0.76 CCL5 (0.40) TDP1ALDH1A1
SCHEMBL5235643 0.74 CHRNB2 (0.53) CCR5ALDH1A1
SCHEMBL5232470 0.73 CCR5 (0.54) CCR5
SCHEMBL5239176 0.72 HTT (0.43) TDP1ALDH1A1
SCHEMBL5240008 0.72 ALDH1A1 (0.48) CCR5ALDH1A1
SCHEMBL5235073 0.72 CHRNB2 (0.53) RIPK1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1761542-A2 OCTAHYDROPYRROLO[3,4-C]PYRROLE DERIVATIVES AN THEIR USE AS ANTIVIRAL AGENTS F.HOFFMANN-LA ROCHE AG (CH) 2007-03-14 EP claimed
WO-2005121145-A2 OCTAHYDRO-PYRROLO[3,4-C] DERIVATIVES AND THEIR USE AS ANTIVIRAL COMPOUNDS F. HOFFMANN-LA ROCHE AG (CH) 2005-12-22 WO claimed