SCHEMBL5263284

SCHEMBL5263284

ClCCn1cnc2c(NC3CCCCC3)nc(Cl)nc21

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 10/20 0.57
ADORA1 P30542 10/20 0.57
ADORA2A P29274 8/20 0.57
CTSL P07711 1/20 0.56
CTSB P07858 1/20 0.56
YTHDC1 Q96MU7 2/20 0.56
ADORA2B P29275 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3451476 0.88 ADORA3 (0.47) ADORA3ADORA1ADORA2ACTSLCTSB
SCHEMBL182902 0.82 ADORA1 (0.63) ADORA3ADORA1ADORA2AYTHDC1ADORA2B
SCHEMBL7442349 0.81 ADORA1 (0.64) ADORA3ADORA1ADORA2AYTHDC1ADORA2B
SCHEMBL17929772 0.80 YTHDC1 (0.63) ADORA3ADORA1ADORA2ACTSLCTSB
SCHEMBL20180099 0.80 CTSL (0.51) ADORA3ADORA1ADORA2ACTSLCTSB
SCHEMBL3451170 0.79 CTSL (0.68) ADORA3ADORA1ADORA2ACTSLCTSB
SCHEMBL17262783 0.78 YTHDC1 (0.61) ADORA3ADORA1ADORA2ACTSLCTSB
SCHEMBL16549253 0.77 YTHDC1 (0.59) ADORA3ADORA1ADORA2AYTHDC1ADORA2B
SCHEMBL13057358 0.75 CDK2 (0.61) ADORA3ADORA1ADORA2AADORA2B
SCHEMBL21348744 0.75 YTHDC1 (0.66) ADORA3ADORA1ADORA2AYTHDC1ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1537111-B1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2007-05-02 EP disclosed
US-20060142575-A1 Hetereoaryl nitrile derivatives NOVARTIS AG (CH) 2006-06-29 US disclosed
EP-1537111-A1 HETEREOARYL NITRILE DERIVATIVES Novartis AG (CH) 2005-06-08 EP disclosed
WO-2004020441-A1 HETEREOARYL NITRILE DERIVATIVES NOVARTIS AG (CH) 2004-03-11 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060142575-A1 Hetereoaryl nitrile derivatives CTSK, CTSZ, CTSE ADORA3 3481/4885ADORA1 3391/4885ADORA2A 3905/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.