SCHEMBL5265221

SCHEMBL5265221

CC(=O)c1ccc(C(F)(F)F)nc1-c1ccccc1.CCOC(=O)c1ccc(C(F)(F)F)nc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
SMN1; SMN2 Q16637 7/20 0.53
RAB9A P51151 6/20 0.53
MAPT P10636 4/20 0.53
NPC1 O15118 4/20 0.53
TP53 P04637 2/20 0.53
LMNA P02545 1/20 0.51
MAPK1 P28482 1/20 0.51
ATM Q13315 1/20 0.51
HSD17B10 Q99714 4/20 0.46
KDM4E B2RXH2 6/20 0.44
MDM2 Q00987 1/20 0.44
HTT P42858 2/20 0.44
TSHR P16473 2/20 0.43
NFKB1 P19838 1/20 0.43
NFKB2 Q00653 1/20 0.43
RELA Q04206 1/20 0.43
CA12 O43570 1/20 0.43
CA9 Q16790 1/20 0.43
MEN1 O00255 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4192118 0.88 ALDH1A1 (0.57) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL1375048 0.85 KDM4E (0.53) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL13853226 0.82 JUN (0.43) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL5260549 0.78 ALDH1A1 (0.47) ALDH1A1SMN1; SMN2MAPTLMNAMAPK1
SCHEMBL5265309 0.77 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL5335693 0.76 L3MBTL1 (0.47) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL13853225 0.74 TUBB4A (0.49) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL22440652 0.74 KDM4E (0.47) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL1007071 0.73 ALDH1A1 (0.51) ALDH1A1SMN1; SMN2RAB9AMAPTNPC1
SCHEMBL1498542 0.72 KDM4E (0.50) ALDH1A1RAB9ANPC1LMNAATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1824828-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS Peakdale Molecular Limited (GB) 2007-08-29 EP disclosed
WO-2006059103-A2 PYRIDINE BASED COMPOUNDS USEFUL AS INTERMEDIATES FOR PHARMACEUTICAL OR AGRICULTURAL END-PRODUCTS PEAKDALE MOLECULAR LIMITED (GB) 2006-06-08 WO disclosed