SCHEMBL5267465

SCHEMBL5267465

CCCCS(=O)(=O)Nc1c[nH]nc1C(=O)NCc1ccccc1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AR P10275 1/20 0.43
TP53 P04637 2/20 0.42
MAPT P10636 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
GAA P10253 3/20 0.41
ALDH1A1 P00352 2/20 0.41
KCNK3 O14649 1/20 0.41
KCNK9 Q9NPC2 1/20 0.41
EPHX2 P34913 1/20 0.41
PARP14 Q460N5 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
PPARG P37231 1/20 0.39
PPARA Q07869 1/20 0.39
POLB P06746 1/20 0.39
PKM P14618 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5267869 0.89 RAB9A (0.47) ARMAPTSMN1; SMN2GAAALDH1A1
SCHEMBL5267514 0.85 F2 (0.46) TP53MAPTSMN1; SMN2GAAALDH1A1
SCHEMBL5265937 0.84 CCNE2 (0.45) ARTP53MAPTSMN1; SMN2ALDH1A1
SCHEMBL5268993 0.84 ALDH1A1 (0.54) TP53MAPTSMN1; SMN2GAAALDH1A1
SCHEMBL5269803 0.83 HPGD (0.48) TP53MAPTSMN1; SMN2ALDH1A1POLB
SCHEMBL5268887 0.81 KCNK3 (0.39) MAPTGAAALDH1A1KCNK3KCNK9
SCHEMBL5265233 0.81 ALDH1A1 (0.44) TP53MAPTSMN1; SMN2GAAALDH1A1
SCHEMBL5268485 0.81 KCNA5 (0.51) TP53MAPTGAAALDH1A1
SCHEMBL5266632 0.81 CASP1 (0.42) TP53MAPTSMN1; SMN2GAAALDH1A1
SCHEMBL5272580 0.80 ALOX15 (0.49) TP53MAPTGAAALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed