SCHEMBL5268887

SCHEMBL5268887

CCCCS(=O)(=O)Nc1c[nH]nc1C(=O)NC

nearest known ligand 0.39

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KCNK3 O14649 1/20 0.39
KCNK9 Q9NPC2 1/20 0.39
HPGD P15428 2/20 0.39
LMNA P02545 1/20 0.39
BRD4 O60885 1/20 0.38
GAA P10253 2/20 0.37
KDM4E B2RXH2 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
PGAM1 P18669 1/20 0.37
BRAF P15056 1/20 0.37
MRGPRX1 Q96LB2 1/20 0.37
PIK3C3 Q8NEB9 1/20 0.36
TRPV1 Q8NER1 1/20 0.36
CCR4 P51679 1/20 0.36
PARP14 Q460N5 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5270110 0.87 KCNK3 (0.42) KCNK3KCNK9HPGDLMNABRD4
SCHEMBL5265937 0.83 CCNE2 (0.45) KCNK3KCNK9KDM4EALDH1A1MAPT
SCHEMBL5268756 0.82 LMNA (0.42) LMNAALDH1A1
SCHEMBL5267465 0.81 AR (0.43) KCNK3KCNK9GAAALDH1A1MAPT
SCHEMBL5267869 0.80 RAB9A (0.47) KCNK3KCNK9HPGDGAAKDM4E
SCHEMBL5267069 0.79 ALDH1A1 (0.39) KCNK3KCNK9HPGDBRD4GAA
SCHEMBL5269803 0.78 HPGD (0.48) HPGDLMNAALDH1A1MAPT
SCHEMBL5271876 0.75 MTNR1A (0.43) GAAALDH1A1
SCHEMBL13816862 0.73 YTHDC1 (0.41) HPGDBRD4KDM4E
SCHEMBL5318573 0.72 SLC40A1 (0.49) HPGDLMNAGAAKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed