SCHEMBL5267757

SCHEMBL5267757

O=C(Cc1ccc(-c2ccccc2)cc1)Nc1c[nH]nc1C(=O)N1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 7/20 0.47
MEN1 O00255 5/20 0.47
KCNQ2 O43526 4/20 0.46
GAA P10253 1/20 0.46
PKM P14618 1/20 0.46
CDK2 P24941 3/20 0.45
CCNE1 P24864 1/20 0.45
CDK9 P50750 1/20 0.45
CDK5 Q00535 1/20 0.45
CDK5R1 Q15078 1/20 0.45
CCNA2 P20248 1/20 0.44
CCNA1 P78396 1/20 0.44
HPGD P15428 1/20 0.44
MAPK1 P28482 1/20 0.44
SLC6A2 P23975 1/20 0.44
SLC6A3 Q01959 1/20 0.44
ALDH1A1 P00352 2/20 0.43
NAAA Q02083 1/20 0.43
CDK1 P06493 1/20 0.42
CDK4 P11802 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5267112 0.82 NPC1 (0.48) KMT2AMEN1GAAHPGDALDH1A1
SCHEMBL5272564 0.81 NPY4R (0.57) GAAMAPK1ALDH1A1LMNANPC1
SCHEMBL5265952 0.80 KMT2A (0.52) KMT2AMEN1GAAPKMCDK2
SCHEMBL5271648 0.80 KMT2A (0.54) KMT2AMEN1PKMCDK2CCNE1
SCHEMBL5266503 0.79 MEN1 (0.61) KMT2AMEN1CDK2CCNE1CDK9
SCHEMBL5270089 0.79 GAA (0.59) KMT2AMEN1GAAPKMMAPK1
SCHEMBL5273651 0.78 HRH3 (0.54) KMT2AMEN1PKMCDK2CCNE1
SCHEMBL5271504 0.78 HPGD (0.53) KMT2AMEN1GAAHPGDALDH1A1
SCHEMBL5268895 0.78 LMNA (0.56) KMT2AMEN1SLC6A2SLC6A3ALDH1A1
SCHEMBL5269971 0.77 L3MBTL1 (0.50) KMT2AMEN1GAAHPGDMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1847531-A1 PYRAZOLE COMPOUND Takeda Pharmaceutical Company Limited (JP) 2007-10-24 EP disclosed