SCHEMBL5307374

SCHEMBL5307374

CCOc1ccccc1N1CCN(CCNC(=O)CN2C(=O)C3CC(O)C(O)CC3C2=O)CC1

nearest known ligand 0.56

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.55
ADRA1D P25100 4/20 0.53
ADRA1A P35348 4/20 0.53
ADRA1B P35368 4/20 0.53
POLB P06746 1/20 0.51
DRD2 P14416 2/20 0.48
DRD3 P35462 1/20 0.48
HTR1A P08908 1/20 0.47
HTR7 P34969 1/20 0.47
DRD4 P21917 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5308285 0.91 DRD2 (0.58) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL5328407 0.90 SLC6A4 (0.55) SLC6A4ADRA1DADRA1AADRA1BPOLB
SCHEMBL5302822 0.89 ADRA1A (0.65) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL5310370 0.86 ADRA1A (0.50) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL6211876 0.84 HTR1A (0.59) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL5325863 0.80 DRD2 (0.59) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL5329403 0.80 ADRA1A (0.65) ADRA1DADRA1AADRA1BDRD2DRD3
Hydrochloric Acid SCHEMBL6211262 0.77 DRD2 (0.54) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL5306802 0.76 ADRA1A (0.49) ADRA1DADRA1AADRA1BDRD2DRD3
SCHEMBL5176069 0.75 HTR1A (0.55) ADRA1DADRA1AADRA1BDRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO claimed
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO disclosed