SCHEMBL5310370

SCHEMBL5310370

O=C(CN1C(=O)C2CC(O)C(O)CC2C1=O)NCCN1CCN(c2ccccc2OC2CCCC2)CC1

nearest known ligand 0.50

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 6/20 0.50
ADRA1D P25100 5/20 0.50
ADRA1B P35368 5/20 0.50
DRD2 P14416 1/20 0.46
DRD3 P35462 1/20 0.46
RAB9A P51151 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5306802 0.90 ADRA1A (0.49) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL5308285 0.87 DRD2 (0.58) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL5302822 0.86 ADRA1A (0.65) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL5307374 0.86 SLC6A4 (0.55) ADRA1AADRA1DADRA1BDRD2DRD3
SCHEMBL4521606 0.85 RAB9A (0.50) ADRA1AADRA1DADRA1BDRD2RAB9A
Hydrochloric Acid SCHEMBL4526875 0.84 RAB9A (0.49) ADRA1AADRA1DADRA1BDRD2RAB9A
SCHEMBL4525015 0.84 HTR1A (0.55) ADRA1AADRA1DADRA1BDRD2DRD3
Hydrochloric Acid SCHEMBL4527605 0.83 HTR1A (0.54) ADRA1AADRA1DADRA1BDRD2DRD3
Phosphoric Acid SCHEMBL5328350 0.82 RAB9A (0.47) ADRA1AADRA1DADRA1BDRD2RAB9A
Succinic Acid SCHEMBL5326107 0.81 RAB9A (0.46) ADRA1AADRA1DADRA1BDRD2RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO claimed
WO-2007029156-A2 ISOINDOLEDIONE DERIVATIVES AS ADRENERGIC RECEPTOR ANTAGONISTS RANBAXY LABORATORIES LIMITED (IN) 2007-03-15 WO disclosed