SCHEMBL5309397

SCHEMBL5309397

COc1cccc(N2N=CCCC2=O)c1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 1/20 0.48
MGLL Q99685 1/20 0.46
MAPT P10636 2/20 0.46
CYP1A2 P05177 1/20 0.43
NPC1 O15118 1/20 0.41
ADRB1 P08588 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.40
PDE4A P27815 1/20 0.40
PDE4B Q07343 1/20 0.40
PDE4C Q08493 1/20 0.40
PDE4D Q08499 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
RAB9A P51151 1/20 0.40
NOTUM Q6P988 1/20 0.40
CTSG P08311 1/20 0.40
CMA1 P23946 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27618946 0.80 KMT2A (0.51) ALOX5MGLLMAPTCYP1A2ADRB1
SCHEMBL10618445 0.77 POLB (0.46) ALOX5MAPTCYP1A2NPC1SMN1; SMN2
SCHEMBL20702773 0.76 CA12 (0.42) PDE4APDE4BPDE4CPDE4D
SCHEMBL20703098 0.72 TUBB4A (0.37) MAPTNPC1PDE4APDE4BPDE4C
SCHEMBL15057788 0.72 HDAC4 (0.46) CYP1A2SMN1; SMN2RAB9A
SCHEMBL27762341 0.72 NPC1 (0.49) ALOX5MGLLMAPTCYP1A2NPC1
SCHEMBL5997170 0.72 MGLL (0.45) MGLLMAPTCYP1A2SMN1; SMN2
SCHEMBL4662941 0.72 MAPT (0.68) MGLLMAPTCYP1A2SMN1; SMN2L3MBTL1
SCHEMBL25366082 0.71 ALOX5 (0.55) ALOX5MGLLMAPTCYP1A2NPC1
SCHEMBL30516650 0.71 ALOX5 (0.55) ALOX5MGLLMAPTCYP1A2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007047394-A2 THIOTRIAZOLYL DERIVATIVES EPIX DELAWARE, INC. (US) 2007-04-26 WO disclosed