SCHEMBL5314570

SCHEMBL5314570

N#Cc1ccc(CNC(=O)CN2CC3CN(CCCc4ccccc4)CC(C2)O3)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 8/20 0.48
HTR2A P28223 3/20 0.48
DRD4 P21917 1/20 0.48
HRH1 P35367 1/20 0.48
OPRM1 P35372 1/20 0.48
DRD2 P14416 7/20 0.46
HTR7 P34969 4/20 0.46
HTR6 P50406 4/20 0.46
HTR5A P47898 1/20 0.46
HTT P42858 3/20 0.45
USP2 O75604 1/20 0.45
KDM4E B2RXH2 1/20 0.45
ALDH1A1 P00352 1/20 0.45
GLA P06280 1/20 0.45
HPGD P15428 1/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
POLB P06746 1/20 0.43
GAA P10253 1/20 0.42
HTR2C P28335 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5316192 0.92 HTT (0.52) HTR1AHTR2ADRD2HTR7HTR6
SCHEMBL5319733 0.90 POLB (0.48) HTR1AHTR2ADRD2HTR7HTR6
SCHEMBL5316933 0.89 KCNH2 (0.47) HTR1AHTR2AHRH1DRD2HTR7
SCHEMBL5319103 0.89 KCNH2 (0.49) HTR1AHRH1DRD2HTR7HTR6
SCHEMBL5315856 0.88 POLB (0.49) HTR1AHTR2ADRD2HTR7HTR6
SCHEMBL5316850 0.88 HTR1A (0.49) HTR1AHTR2ADRD4HRH1OPRM1
SCHEMBL5319026 0.88 HTR1A (0.49) HTR1AHTR2ADRD4HRH1OPRM1
SCHEMBL5314874 0.87 POLB (0.54) HTR1AHTR2ADRD2HTR7HTR6
SCHEMBL5315877 0.86 ABCB1 (0.48) HTR1AHTR2ADRD4HRH1OPRM1
SCHEMBL5315867 0.85 ERCC1 (0.44) DRD2HTTUSP2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO claimed
WO-2007069986-A1 NEW OXABISPIDINE COMPOUNDS FOR THE TREATMENT OF CARDIAC ARRHYTHMIAS ASTRAZENECA AB (SE) 2007-06-21 WO disclosed