SCHEMBL5314853

SCHEMBL5314853

COc1cc2c(cc1C)CC(N)C2

nearest known ligand 0.48

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADRA1A P35348 2/20 0.48
FYN P06241 1/20 0.43
DRD2 P14416 2/20 0.42
DRD3 P35462 2/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CYP3A4 P08684 1/20 0.41
MAPT P10636 1/20 0.41
ALDH1A1 P00352 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ALOX15 P16050 1/20 0.40
MAPK1 P28482 1/20 0.40
TAAR1 Q96RJ0 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3041826 0.87 ADRA1A (0.56) ADRA1AFYNDRD2DRD3CA1
Hydrochloric Acid SCHEMBL1788805 0.85 ADRA1A (0.54) ADRA1AFYNDRD2DRD3CA1
SCHEMBL17014922 0.82 CYP3A4 (0.43) CA1CA2CYP3A4MAPTALDH1A1
SCHEMBL4388677 0.80 FYN (0.56) ADRA1AFYNDRD2DRD3CA1
SCHEMBL16816267 0.78 ADRA1A (0.47) ADRA1AFYNDRD2DRD3CA1
SCHEMBL17014945 0.77 MEN1 (0.41) CA1CA2CYP3A4MAPTALDH1A1
SCHEMBL22953307 0.76 MAPT (0.71) DRD2DRD3CYP3A4MAPTALDH1A1
SCHEMBL12595457 0.76 MAPT (0.71) DRD2DRD3CYP3A4MAPTALDH1A1
SCHEMBL7339771 0.74 DRD2 (0.62) ADRA1ADRD2DRD3MAPTALDH1A1
SCHEMBL8765937 0.74 DRD2 (0.62) ADRA1ADRD2DRD3MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 81 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES INC (US) 2025-11-27 US claimed
EP-4618980-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES Freedom Biosciences, Inc. (US) 2025-09-24 EP claimed
WO-2024107445-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES, INC. (US) 2024-05-23 WO claimed
CN-112270066-B Optimization method for calculating rigid coupling coefficient of satellite and computer equipment 航天科工空间工程发展有限公司 2022-04-19 CN claimed
WO-2007069925-A2 NON-NEUROTOXIC RECREATIONAL DRUGS AND A METHOD OF TREATING RECREATIONAL DRUG ABUSE STARGATE INTERNATIONAL LIMITED (NZ) 2007-06-21 WO claimed
WO-2026107229-A1 REDUCING THE ADDICTIVE LIABILITY OF OPIOID ANALGESICS BY CO- ADMINISTERING 5HT2 RECEPTOR AGONISTS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2026-05-21 WO disclosed
WO-2026099114-A1 POWER SUPPLY SYSTEM WITH HETEROGENEOUS POWER SUPPLIES FOR AUTOMATIC PARALLEL OPERATION PHOENIX CONTACT GMBH & CO. KG (DE) 2026-05-15 WO disclosed
US-20260135486-A1 RIPPLE SUPPRESSION IN MULTI-PHASE BUCK CONVERTERS MAXLINEAR, INC. (US) 2026-05-14 US disclosed
EP-4713342-A2 SYSTEMS AND METHODS FOR REGULATING TARGET GENES Epicrispr Biotechnologies, Inc. (US) 2026-03-25 EP disclosed
US-20260049109-A1 NOVEL IMMUNOMODULATORY, NEUROMODULATORY, OSTEOGENIC, AND ANTI-OSTEOPOROTIC HKUOT-S2 PROTEIN THAT ENHANCES BONE FRACTURE REPAIRS AND SUPPRESSES OSTEOPOROSIS DEVELOPMENT UNIV HONG KONG (HK) 2026-02-19 US disclosed
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES FREEDOM BIOSCIENCES INC (US) 2025-11-27 US disclosed
EP-4618980-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES Freedom Biosciences, Inc. (US) 2025-09-24 EP disclosed
US-20110224263-A1 Cyclic pyridyl-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals SANOFI-AVENTIS (FR) 2011-09-15 US disclosed
WO-2009080223-A1 CYCLIC PYRIDYL-N-(1,3,4)-THIADIAZOL-2-YL-BENZENE SULFONAMIDES, PROCESSES FOR THEIR PREPARATION AND THEIR USE AS PHARMACEUTICALS SANOFI-AVENTIS (FR) 2009-07-02 WO disclosed
WO-2007069925-A2 NON-NEUROTOXIC RECREATIONAL DRUGS AND A METHOD OF TREATING RECREATIONAL DRUG ABUSE STARGATE INTERNATIONAL LIMITED (NZ) 2007-06-21 WO disclosed
WO-2007069925-A2 NON-NEUROTOXIC RECREATIONAL DRUGS AND A METHOD OF TREATING RECREATIONAL DRUG ABUSE STARGATE INTERNATIONAL LIMITED (NZ) 2007-06-21 WO disclosed
US-20040005347-A1 Composition comprising cocoa N. V. NUTRICIA (NL) 2004-01-08 US disclosed
EP-1370273-A1 COMPOSITION COMPRISING COCOA AND A DOPAMINE D2 RECEPTOR AGONIST N.V. Nutricia (NL) 2003-12-17 EP disclosed
US-20020172732-A1 Composition comprising cocoa GENERAL NUTRITION INVESTMENT COMPANY 2002-11-21 US disclosed
WO-2002074321-A1 COMPOSITION COMPRISING COCOA AND A DOPAMINE D2 RECEPTOR AGONIST N.V. NUTRICIA (NL) 2002-09-26 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250360137-A1 ENHANCEMENT OF THE EFFICACY OF SEROTONERGIC PSYCHEDELIC DRUGS IN THE TREATMENT OR PREVENTION OF CERTAIN NEUROPSYCHIATRIC DISORDERS THROUGH INHIBITION OF TYPE-9 PHOSPHODIESTERASES PDE9A, PDE3A, PDE2A ADRA1A 177/4885FYN 3215/4885DRD2 123/4885
US-20260049109-A1 NOVEL IMMUNOMODULATORY, NEUROMODULATORY, OSTEOGENIC, AND ANTI-OSTEOPOROTIC HKUOT-S2 PROTEIN THAT ENHANCES BONE FRACTURE REPAIRS AND SUPPRESSES OSTEOPOROSIS DEVELOPMENT SOST, IRF3, BMP2 ADRA1A 3362/4885FYN 2914/4885DRD2 4610/4885
US-20110224263-A1 Cyclic pyridyl-N-[1,3,4]-thiadiazol-2-yl-benzene sulfonamides, processes for their preparation and their use as pharmaceuticals PPARD, PPARG, PPARA ADRA1A 451/4885FYN 2183/4885DRD2 1887/4885
US-20260135486-A1 RIPPLE SUPPRESSION IN MULTI-PHASE BUCK CONVERTERS DSP, RIPK1, DNER ADRA1A 4178/4885FYN 3745/4885DRD2 115/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.