SCHEMBL5314922

SCHEMBL5314922

CNc1cc(-c2ccc(F)cc2F)c2nc(Nc3ccc(CN4CC(C)OC(C)C4)cn3)sc2n1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1B Q01064 2/20 0.35
GRM2 Q14416 2/20 0.34
S1PR1 P21453 4/20 0.34
S1PR3 Q99500 3/20 0.34
CNR2 P34972 1/20 0.34
GRIN2B Q13224 1/20 0.33
CDK4 P11802 5/20 0.33
CCND3 P30281 4/20 0.33
CDK6 Q00534 4/20 0.33
CDK1 P06493 3/20 0.33
MET P08581 1/20 0.33
MERTK Q12866 1/20 0.33
HTR2A P28223 1/20 0.33
CCNA2 P20248 3/20 0.32
DYRK2 Q92630 2/20 0.32
CCND1 P24385 2/20 0.32
TRPV1 Q8NER1 1/20 0.32
CCNT1 O60563 1/20 0.32
CDK2 P24941 1/20 0.32
CDK7 P50613 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5315261 0.87 BDKRB1 (0.37) CNR2GRIN2BCDK4CCND3CDK6
SCHEMBL5311867 0.86 MERTK (0.45) CDK4CCND3CDK6CDK1MET
SCHEMBL5313507 0.86 DYRK2 (0.45) CDK4CCND3CDK6CDK1MET
SCHEMBL5336063 0.85 GRM2 (0.37) GRM2CNR2CDK4CCND3CDK6
SCHEMBL5315552 0.78 BDKRB1 (0.40) GRM2CNR2CDK4CCND3CDK6
SCHEMBL5311883 0.77 TNIK (0.45) GRM2CDK4CCND3CDK6CDK1
SCHEMBL5314023 0.76 KDR (0.47) CDK1METMERTKCDK2CDK9
SCHEMBL5333911 0.76 MERTK (0.38) GRM2METMERTKTRPV1CCNT1
SCHEMBL5334782 0.75 MERTK (0.43) METMERTK
SCHEMBL5312754 0.73 DYRK2 (0.49) CDK4CCND3CDK6CCNA2DYRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO claimed
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO disclosed