SCHEMBL5336063

SCHEMBL5336063

CNc1cc(-c2ccc(F)cc2F)c2nc(Nc3ccc(CN4CCC(N(C)C)C4)cn3)sc2n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM2 Q14416 1/20 0.37
MAP4K4 O95819 2/20 0.37
SCN1A P35498 6/20 0.36
SCN8A Q9UQD0 6/20 0.36
CDK4 P11802 3/20 0.36
CCND1 P24385 2/20 0.36
CCNT1 O60563 2/20 0.36
CDK9 P50750 2/20 0.36
TNIK Q9UKE5 1/20 0.35
CDK6 Q00534 2/20 0.35
FLT3 P36888 1/20 0.35
MERTK Q12866 1/20 0.35
GAS6 Q14393 1/20 0.35
CNR2 P34972 1/20 0.34
PDGFRB P09619 2/20 0.34
KDR P35968 2/20 0.34
MELK Q14680 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCND3 P30281 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5311867 0.85 MERTK (0.45) CDK4TNIKCDK6MERTKCCNA2
SCHEMBL5314922 0.85 PDE1B (0.35) GRM2CDK4CCND1CCNT1CDK9
SCHEMBL5313507 0.85 DYRK2 (0.45) CDK4CCND1CDK6MERTKKDR
SCHEMBL5315261 0.85 BDKRB1 (0.37) CDK4CCND1CCNT1CDK9CDK6
SCHEMBL14531378 0.78 MELK (0.39) GRM2MAP4K4SCN1ASCN8ACDK4
SCHEMBL5333911 0.76 MERTK (0.38) GRM2MAP4K4CCNT1CDK9FLT3
SCHEMBL5311883 0.76 TNIK (0.45) GRM2CDK4TNIKCDK6MERTK
SCHEMBL5315552 0.75 BDKRB1 (0.40) GRM2CDK4CCND1CDK6CNR2
SCHEMBL5331801 0.75 MAP4K4 (0.38) GRM2MAP4K4SCN1ASCN8AMELK
SCHEMBL5334782 0.74 MERTK (0.43) MERTKKDR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007058482-A1 NOVEL INHIBITORS OF PROTEIN KINASE LG LIFE SCIENCES, LTD. (KR) 2007-05-24 WO claimed