SCHEMBL5327640

SCHEMBL5327640

CC(C)(C)OC(=O)C1=CCN(Cc2ccccc2)C1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
KMT2A Q03164 3/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.41
NPFFR1 Q9GZQ6 1/20 0.40
NPFFR2 Q9Y5X5 1/20 0.40
ACHE P22303 2/20 0.40
MEN1 O00255 1/20 0.40
OPRM1 P35372 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
SIRT2 Q8IXJ6 1/20 0.38
SIRT1 Q96EB6 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7534318 0.85 MEN1 (0.47) KMT2AALDH1A1LMNAACHEMEN1
SCHEMBL3222039 0.82 LMNA (0.48) KMT2AALDH1A1LMNAMEN1
SCHEMBL1344511 0.80 CYP2D6 (0.46) KMT2AALDH1A1LMNAACHESIGMAR1
SCHEMBL28039452 0.79 SIGMAR1 (0.47) KMT2AALDH1A1LMNAL3MBTL1MEN1
SCHEMBL20314913 0.79 ALDH1A1 (0.42) KMT2AALDH1A1LMNAMEN1SIGMAR1
SCHEMBL6640189 0.71 LMNA (0.54) KMT2AALDH1A1LMNAMEN1
SCHEMBL3079800 0.71 MEN1 (0.48) KMT2AALDH1A1MEN1
SCHEMBL14087069 0.71 DRD2 (0.47) KMT2AALDH1A1LMNAL3MBTL1NPFFR1
SCHEMBL25173575 0.70 S1PR5 (0.56) KMT2AALDH1A1LMNAL3MBTL1
SCHEMBL2862442 0.70 ALDH1A1 (0.60) KMT2AALDH1A1LMNAL3MBTL1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12465590-B2 Oxalamido-substituted tricyclic inhibitors of hepatitis b virus OSPEDALE SAN RAFFAELE S.R.L. (IT) 2025-11-11 US disclosed
CN-119409710-A Oxamide substituted hepatitis b virus tricyclic inhibitors 圣拉斐尔医院有限公司 2025-02-11 CN disclosed
CN-114555608-B Oxamide substituted hepatitis b virus tricyclic inhibitors 圣拉斐尔医院有限公司 2024-11-01 CN disclosed
US-20220241241-A1 OXALAMIDO-SUBSTITUTED TRICYCLIC INHIBITORS OF HEPATITIS B VIRUS ISTITUTO NAZIONALE DI GENETICA MOLECOLARE - INGM (IT) 2022-08-04 US disclosed
CN-114555608-A Oxamide substituted tricyclic inhibitors of hepatitis b virus 分子遗传国家研究所(INGM) 2022-05-27 CN disclosed
EP-3972979-A1 OXALAMIDO-SUBSTITUTED TRICYCLIC INHIBITORS OF HEPATITIS B VIRUS Antios Therapeutics, Inc. (US) 2022-03-30 EP disclosed
WO-2020234483-A1 OXALAMIDO-SUBSTITUTED TRICYCLIC INHIBITORS OF HEPATITIS B VIRUS ISTITUTO NAZIONALE DI GENETICA MOLECOLARE - INGM (IT) 2020-11-26 WO disclosed
WO-2007034406-A1 PYRROLIDINE-3-CARBOXYLIC ACID AMIDE DERIVATIVES AND THEIR USE AS INHIBITORS OF RENIN ACTELION PHARMACEUTICALS LTD (CH) 2007-03-29 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12465590-B2 Oxalamido-substituted tricyclic inhibitors of hepatitis b virus OAT, SLC10A1, OTC CRHBP 4297/4885CRHR2 4819/4885KMT2A 3220/4885
US-20220241241-A1 OXALAMIDO-SUBSTITUTED TRICYCLIC INHIBITORS OF HEPATITIS B VIRUS OAT, OTC, SLC10A1 CRHBP 4112/4885CRHR2 4848/4885KMT2A 3235/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.