SCHEMBL5333327

SCHEMBL5333327

C=CCc1c(N)c(CC=C)c(CC=C)c(-c2ccc(N)cc2)c1CC=C

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.37
CYP3A4 P08684 2/20 0.37
TDP1 Q9NUW8 2/20 0.37
TP53 P04637 1/20 0.37
GABRA1 P14867 1/20 0.36
GABRB2 P47870 1/20 0.36
MAPT P10636 3/20 0.33
HPGD P15428 2/20 0.33
GAA P10253 1/20 0.33
KDM4E B2RXH2 1/20 0.33
RAB9A P51151 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
IMPDH2 P12268 1/20 0.33
TAAR1 Q96RJ0 1/20 0.32
HSD17B10 Q99714 1/20 0.32
AKR1B1 P15121 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
APP P05067 1/20 0.30
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10885436 0.98 ALDH1A1 (0.36) ALDH1A1CYP3A4TDP1TP53GABRA1
SCHEMBL28716719 0.76 NPSR1 (0.38) ALDH1A1IMPDH2
SCHEMBL1334154 0.72 IMPDH2 (0.41) ALDH1A1CYP3A4TDP1TP53GABRA1
SCHEMBL324128 0.72 HPGD (0.37) ALDH1A1CYP3A4TDP1MAPTHPGD
SCHEMBL3423968 0.71 NPSR1 (0.35) ALDH1A1IMPDH2
SCHEMBL7596717 0.69 TDP1 (0.42) ALDH1A1CYP3A4TDP1TP53MAPT
SCHEMBL29129796 0.69 CYP3A4 (0.42) ALDH1A1CYP3A4TDP1TP53MAPT
SCHEMBL6013231 0.69 GABRA1 (0.44) GABRA1GABRB2MAPTGAASMN1; SMN2
SCHEMBL716339 0.68 ALDH1A1 (0.52) ALDH1A1CYP3A4TDP1TP53GABRA1
Benzidine SCHEMBL28789348 0.67 CYP3A4 (0.54) ALDH1A1CYP3A4TDP1TP53MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 79 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0918881-B1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND AMIRA MEDICAL (US) 2004-02-11 EP claimed
WO-2000039586-A2 TETRAMETHYLBENZIDINE FORMULATION FOR HORSERADISH PEROXIDASE ENZYME ASSAYS SEDUM LABORATORIES (US) 2000-07-06 WO claimed
EP-0918881-A1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND Mercury Diagnostics Inc. (US) 1999-06-02 EP claimed
US-5824491-A OXIDASE ENZYME AS ANALYTE ON SUBSTRATE, FORMING PEROXIDE, BENZIDINE DYE PRECURSOR, PEROXIDASE ENZYME WITH ANTIPYRENE COMPOUND MERCURY DIAGNOSTICS, INC. (US) 1998-10-20 US claimed
WO-1997044482-A1 DRY REAGENT TEST STRIP COMPRISING BENZIDINE DYE PRECURSOR AND ANTIPYRINE COMPOUND MERCURY DIAGNOSTICS INC. (US) 1997-11-27 WO claimed
US-5610026-A OF AN AQUEOUS SOLUTION CONTAINING A TETRAALKYLBENZIDINE OR A SALT THEREOF, A PEROXIDE OR A SYSTEM GENERATING HYDROGEN PEROXIDE AND A BUFFER BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1997-03-11 US claimed
US-5491094-A COLORIMETRIC ANALYSIS INDICATOR 3,3*,5,5*-TETRAALKYLBENZIDINE INDUSTRIAL TEST SYSTEMS, INC. (US) 1996-02-13 US claimed
US-5206150-A Tetramethylbenzidine, peroxide and bacitracin as stabilizer; incubation UNIVERSITY OF KENTUCKY RESEARCH FOUNDATION (US) 1993-04-27 US claimed
EP-0224813-B1 MEANS FOR DETECTING PEROXIDASE ACTIVITY WITH A STABILIZER, PREPARATION PROCESS AND ITS USE BEHRINGWERKE Aktiengesellschaft (DE) 1990-09-26 EP claimed
EP-0224210-B1 MEANS FOR DETECTING PEROXIDASE ACTIVITY, PREPARATION PROCESS AND ITS USE BEHRINGWERKE Aktiengesellschaft (DE) 1990-08-29 EP claimed
US-4891314-A STORAGE STABILITY BEHRINGWERKE AKTIENGESELLSCHAFT (DE) 1990-01-02 US claimed
US-4562148-A IMMUNOASSAY, CARBOXYLATE OR SULFONATE POLYMER MILES LABORATORIES, INC. (US) 1985-12-31 US claimed
JP-1104196-A None JP disclosed
JP-8080199-A None JP disclosed
JP-61052300-A None JP disclosed
JP-8313525-A None JP disclosed
US-4385114-A DETERMINATION OF HYDROGEN PEROXIDE OR PEROXIDASE BOEHRINGER MANNHEIM GMBH (DE) 1983-05-24 US disclosed
EP-0078965-A1 Method for preparing an analytical element preventing reagent migration MILES LABORATORIES, INC. (US) 1983-05-18 EP disclosed
EP-0071934-A1 Method for preparing a color stable chromogenic analytical element MILES LABORATORIES, INC. (US) 1983-02-16 EP disclosed
US-4361648-A POLYMERIC MORDANT, TETRAALKYLBENZIDINE HYDROCHLORIDE, ENZYME, PEROXIDATIVELY ACTIVE MATERIAL MILES LABORATORIES, INC. (US) 1982-11-30 US disclosed