SCHEMBL5339306

SCHEMBL5339306

CC(C)CNC(=O)c1ccc(-c2ccc(C(=O)c3cc(F)ccc3C(F)(F)F)nc2)nn1

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SCD O00767 5/20 0.41
GABRA1 P14867 1/20 0.40
DYRK1A Q13627 1/20 0.37
GRIN2B Q13224 1/20 0.37
HDAC4 P56524 1/20 0.36
GCGR P47871 3/20 0.36
NPC1 O15118 4/20 0.36
RAB9A P51151 4/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 2/20 0.35
HPGD P15428 1/20 0.35
POLB P06746 1/20 0.35
STING1 Q86WV6 1/20 0.35
ROCK2 O75116 1/20 0.35
PRKG1 Q13976 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5310783 0.89 SCD (0.46) SCDGABRA1
SCHEMBL5312928 0.84 SCD (0.50) SCDGABRA1
SCHEMBL5307870 0.82 ASPH (0.43) SCDALDH1A1STING1
SCHEMBL5315830 0.73 ASPH (0.48)
SCHEMBL5312220 0.72 SCD (0.47) SCDGABRA1
SCHEMBL5376686 0.71 NPC1 (0.39) SCDNPC1ALDH1A1STING1
SCHEMBL5310095 0.70 KCNMA1 (0.48) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL13932843 0.70 MLYCD (0.48) HDAC4SMN1; SMN2ALDH1A1HSD17B10LMNA
SCHEMBL5314293 0.69 ADORA2A (0.47) NPC1RAB9ASMN1; SMN2ALDH1A1LMNA
SCHEMBL5313162 0.69 CNR2 (0.48) SCDLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044085-A2 HETEROARYL COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-19 WO disclosed