SCHEMBL5376686

SCHEMBL5376686

O=C(O)c1ccc(-c2ccc(C(=O)c3cc(F)ccc3C(F)(F)F)cc2)nn1

nearest known ligand 0.39

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.39
RXFP1 Q9HBX9 1/20 0.39
CYP2C8 P10632 1/20 0.39
KMO O15229 2/20 0.39
KDM4E B2RXH2 1/20 0.38
ALDH1A1 P00352 1/20 0.38
SCD O00767 4/20 0.38
LDHA P00338 1/20 0.36
KIF11 P52732 1/20 0.35
ASPH Q12797 1/20 0.35
DHODH Q02127 1/20 0.34
STING1 Q86WV6 1/20 0.34
EIF4E P06730 1/20 0.34
PTPRB P23467 1/20 0.34
BCL2L1 Q07817 1/20 0.34
BAD Q92934 1/20 0.34
EPRS1 P07814 1/20 0.34
CHRNA7 P36544 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5307870 0.88 ASPH (0.43) KMOKDM4EALDH1A1SCDASPH
SCHEMBL5307717 0.83 ASPH (0.45) KMOKIF11ASPHBCL2L1BAD
SCHEMBL5315830 0.77 ASPH (0.48) KMOASPH
SCHEMBL5313162 0.74 CNR2 (0.48) KMOSCDASPH
SCHEMBL28021530 0.72 CES2 (0.50) ALDH1A1KIF11
SCHEMBL5339306 0.71 SCD (0.41) NPC1ALDH1A1SCDSTING1
SCHEMBL5312928 0.71 SCD (0.50) SCD
SCHEMBL29406303 0.70 KEAP1 (0.55) KDM4EALDH1A1ASPH
SCHEMBL222474 0.70 KEAP1 (0.55) KDM4EALDH1A1ASPH
SCHEMBL5310364 0.68 CNR2 (0.47) KMOASPH

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2007044085-A2 HETEROARYL COMPOUNDS AND THEIR USES AS THERAPEUTIC AGENTS XENON PHARMACEUTICALS INC. (CA) 2007-04-19 WO disclosed