SCHEMBL535076

SCHEMBL535076

O=C(Nc1ccccc1N1CCc2ccccc21)[C@@H]1CC[C@@H]1CO

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNQ2 O43526 1/20 0.44
MAPT P10636 5/20 0.41
LMNA P02545 2/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TSHR P16473 3/20 0.39
P2RY1 P47900 2/20 0.39
ALDH1A1 P00352 3/20 0.39
GAA P10253 1/20 0.39
MAPK1 P28482 1/20 0.39
HSD17B10 Q99714 1/20 0.39
SMN1; SMN2 Q16637 3/20 0.38
KMT2A Q03164 1/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
TP53 P04637 1/20 0.38
PKM P14618 1/20 0.38
NFKB1 P19838 1/20 0.38
NFKB2 Q00653 1/20 0.38
RELA Q04206 1/20 0.38
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11445291 0.81 TSHR (0.52) KCNQ2MAPTLMNANPSR1TSHR
SCHEMBL11446797 0.79 ALDH1A1 (0.56) KCNQ2LMNANPSR1TSHRP2RY1
SCHEMBL11445341 0.78 TSHR (0.62) KCNQ2LMNANPSR1TSHRALDH1A1
SCHEMBL11445874 0.74 ALDH1A1 (0.64) MAPTLMNAP2RY1ALDH1A1SMN1; SMN2
SCHEMBL11453386 0.72 RAB9A (0.53) KCNQ2MAPTLMNANPSR1TSHR
SCHEMBL11446342 0.71 SMN1; SMN2 (0.59) MAPTLMNANPSR1TSHRALDH1A1
SCHEMBL11445253 0.71 KCNQ2 (0.65) KCNQ2MAPTLMNANPSR1TSHR
SCHEMBL535321 0.70 L3MBTL1 (0.56) MAPTLMNAALDH1A1GAASMN1; SMN2
SCHEMBL8938751 0.70 MAPT (0.47) MAPTTSHRP2RY1ALDH1A1GAA
SCHEMBL10623856 0.69 KDM4E (0.58) MAPTALDH1A1HSD17B10SMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2414323-A1 DERIVATIVES OF AMINOCYCLOBUTANE OR AMINOCYCLOBUTENE, THEIR METHOD OF PREPARATION AND THEIR USE AS MEDICAL PRODUCTS Pierre Fabre Médicament (FR) 2012-02-08 EP disclosed
WO-2010112597-A1 DERIVATIVES OF AMINOCYCLOBUTANE OR AMINOCYCLOBUTENE, THEIR METHOD OF PREPARATION AND THEIR USE AS MEDICAL PRODUCTS PIERRE FABRE MEDICAMENT (FR) 2010-10-07 WO disclosed