SCHEMBL5353450

SCHEMBL5353450

CC(C)(N)CCn1cnc(-c2ccccc2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE10A Q9Y233 1/20 0.44
HPGDS O60760 1/20 0.43
CYP2E1 P05181 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2A6 P11509 2/20 0.43
CYP2C9 P11712 2/20 0.43
CYP2B6 P20813 2/20 0.43
CYP2C19 P33261 2/20 0.43
CYP2D6 P10635 1/20 0.43
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
NLRP3 Q96P20 1/20 0.38
LMNA P02545 2/20 0.36
MAPT P10636 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
ALDH1A1 P00352 1/20 0.36
HTT P42858 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
PLK4 O00444 1/20 0.36
JAK2 O60674 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2198329 0.85 RAB9A (0.38) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
Ammonia Solution, Strong SCHEMBL2287120 0.84 RAB9A (0.37) CYP2E1CYP3A4CYP2A6CYP2C9CYP2B6
SCHEMBL2199232 0.83 MAPT (0.48) NPC1RAB9ALMNAMAPTALDH1A1
SCHEMBL4890520 0.80 FABP4 (0.44) LMNAMAPT
SCHEMBL7990801 0.79 CYP2E1 (0.53) PDE10AHPGDSCYP2E1CYP3A4CYP2A6
Hydrochloric Acid SCHEMBL28812335 0.78 PDE10A (0.48) PDE10AHPGDSCYP2E1CYP3A4CYP2A6
SCHEMBL2910946 0.77 CYP2E1 (0.67) PDE10AHPGDSCYP2E1CYP3A4CYP2A6
SCHEMBL5924494 0.76 PDE10A (0.47) PDE10AHPGDSCYP2E1CYP3A4CYP2A6
SCHEMBL651699 0.76 CYP2E1 (0.50) PDE10AHPGDSCYP2E1CYP3A4CYP2A6
SCHEMBL12985062 0.76 CYP2E1 (0.42) PDE10AHPGDSCYP2E1CYP3A4CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7214698-B2 Beta-agonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2007-05-08 US disclosed
US-20060173061-A1 New beta-agonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2006-08-03 US disclosed
US-20040127733-A1 New beta-agonists, processes for preparing them and their use as pharmaceutical compositions BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2004-07-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20060173061-A1 New beta-agonists, processes for preparing them and their use as pharmaceutical compositions ADRB1, ADRB2, ADRA1A PDE10A 101/4885HPGDS 1243/4885CYP2E1 511/4885
US-20040127733-A1 New beta-agonists, processes for preparing them and their use as pharmaceutical compositions ADRB1, ADRA1A, ADRA1D PDE10A 86/4885HPGDS 1194/4885CYP2E1 473/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.