SCHEMBL5371873

SCHEMBL5371873

Cc1nc(-c2ccc(F)cc2)c(-c2ccc(F)cc2)[nH]1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.67
HPGD P15428 2/20 0.67
SMN1; SMN2 Q16637 2/20 0.67
MAPK14 Q16539 12/20 0.56
MAPK13 O15264 10/20 0.56
MAPK12 P53778 10/20 0.56
MAPK11 Q15759 10/20 0.56
GCGR P47871 9/20 0.56
GSK3B P49841 3/20 0.56
PRKD3 O94806 2/20 0.56
MAP4K4 O95819 2/20 0.56
FRK P42685 2/20 0.56
MAPK9 P45984 2/20 0.56
CSNK1A1 P48729 2/20 0.56
CSNK1D P48730 2/20 0.56
PRKD2 Q9BZL6 2/20 0.56
CLK4 Q9HAZ1 2/20 0.56
PTK6 Q13882 1/20 0.56
BRAF P15056 1/20 0.54
PTGS1 P23219 2/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7090083 0.89 MAPK14 (0.65) KDM4EHPGDSMN1; SMN2MAPK14MAPK13
SCHEMBL7083972 0.86 PTGS2 (0.75) SMN1; SMN2MAPK14MAPK11CSNK1A1CSNK1D
SCHEMBL7087818 0.85 ALOX5 (0.65) KDM4EHPGDSMN1; SMN2MAPK14MAPK11
SCHEMBL15676793 0.85 MAPK14 (0.50) KDM4EHPGDSMN1; SMN2MAPK14MAPK13
SCHEMBL16713033 0.82 KDM4E (0.44) KDM4EHPGDSMN1; SMN2MAPK14MAPK13
SCHEMBL18041684 0.82 TGFBR1 (0.53) KDM4EHPGDSMN1; SMN2MAPK14MAPK13
SCHEMBL7041734 0.81 KDM4E (0.67) KDM4EHPGDSMN1; SMN2MAPK14MAPK13
SCHEMBL3371979 0.80 MAPK14 (0.74) KDM4EHPGDSMN1; SMN2MAPK14MAPK13
SCHEMBL1068923 0.80 KDM4E (1.00) KDM4EHPGDSMN1; SMN2MAPK14MAPK13
SCHEMBL18041867 0.80 MAPK14 (0.54) KDM4EHPGDSMN1; SMN2MAPK14MAPK13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE39634-E1 Bisarylimidazoly fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-15 US disclosed
US-RE39634-E1 Bisarylimidazoly fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-15 US disclosed
US-RE39634-E1 Bisarylimidazoly fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY (US) 2007-05-15 US disclosed
EP-1389107-A4 BISARYLIMIDAZOLYL FATTY ACID AMIDE HYDROLASE INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2005-10-12 EP disclosed
EP-1389107-A1 BISARYLIMIDAZOLYL FATTY ACID AMIDE HYDROLASE INHIBITORS Bristol-Myers Squibb Company (US) 2004-02-18 EP disclosed
US-6562846-B2 Bisarylimidazolyl fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2003-05-13 US disclosed
US-20020188009-A1 Bisarylimidazolyl fatty acid amide hydrolase inhibitors BRISTOL-MYERS SQUIBB COMPANY 2002-12-12 US disclosed
WO-2002087569-A1 BISARYLIMIDAZOLYL FATTY ACID AMIDE HYDROLASE INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2002-11-07 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020188009-A1 Bisarylimidazolyl fatty acid amide hydrolase inhibitors FAAH, FAAH2, FASN KDM4E 2584/4885HPGD 510/4885SMN1; SMN2 4026/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.