SCHEMBL5467189

SCHEMBL5467189

COC(=O)c1ccccc1NS(=O)(=O)c1cccc([N+](=O)[O-])c1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DDX3X O00571 1/20 0.66
CYP3A4 P08684 1/20 0.62
CYP2C9 P11712 1/20 0.62
RECQL P46063 1/20 0.62
MEN1 O00255 2/20 0.61
KMT2A Q03164 2/20 0.61
GAA P10253 1/20 0.61
MAPT P10636 2/20 0.56
LMNA P02545 2/20 0.55
MAPK1 P28482 1/20 0.55
NFKBIA P25963 1/20 0.55
RELA Q04206 1/20 0.55
ALDH1A1 P00352 3/20 0.54
CA1 P00915 1/20 0.54
CA2 P00918 1/20 0.54
MMP1 P03956 1/20 0.54
MMP2 P08253 1/20 0.54
MMP9 P14780 1/20 0.54
MMP8 P22894 1/20 0.54
MMP13 P45452 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3279892 0.88 LMNA (0.59) CYP3A4CYP2C9MEN1KMT2AGAA
SCHEMBL5467045 0.85 DDX3X (0.69) DDX3XCYP3A4CYP2C9RECQLMEN1
SCHEMBL3983832 0.84 HPGD (0.65) DDX3XCYP3A4CYP2C9MEN1KMT2A
SCHEMBL5468786 0.81 ALDH1A1 (0.71) DDX3XMEN1KMT2AMAPTLMNA
SCHEMBL26931604 0.81 GUSB (0.63) CYP3A4CYP2C9MEN1KMT2AGAA
SCHEMBL13011714 0.80 KMT2A (0.74) CYP3A4CYP2C9MEN1KMT2AGAA
SCHEMBL23200347 0.80 KEAP1 (0.65) MEN1KMT2AGAALMNAMAPK1
SCHEMBL5467385 0.80 DDX3X (0.71) DDX3XMEN1KMT2AMAPTLMNA
SCHEMBL11863940 0.80 DDX3X (1.00) DDX3XCYP3A4CYP2C9RECQLMEN1
SCHEMBL7373349 0.79 KMT2A (0.68) CYP3A4CYP2C9MEN1KMT2AGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10933038-B2 Use of (benzenesulfonamido) benzamide compounds for inhibiting liver fibrosis Hebei Medfaith Pharmaceutical Technology Co., Ltd. (CN) 2021-03-02 US disclosed
US-10933038-B2 Use of (benzenesulfonamido) benzamide compounds for inhibiting liver fibrosis Hebei Medfaith Pharmaceutical Technology Co., Ltd. (CN) 2021-03-02 US disclosed
US-20190274979-A2 USE OF (BENZENESULFONAMIDO)BENZAMIDE COMPOUNDS FOR INHIBITING LIVER FIBROSIS Hebei Medfaith Pharmaceutical Technology Co., Ltd. (CN) 2019-09-12 US disclosed
US-20190274979-A2 USE OF (BENZENESULFONAMIDO)BENZAMIDE COMPOUNDS FOR INHIBITING LIVER FIBROSIS Hebei Medfaith Pharmaceutical Technology Co., Ltd. (CN) 2019-09-12 US disclosed
US-20180333376-A1 USE OF (BENZENESULFONAMIDO) BENZAMIDE COMPOUNDS FOR INHIBITING LIVER FIBROSIS Hebei Medfaith Pharmaceutical Technology Co., Ltd. (CN) 2018-11-22 US disclosed
US-20070010537-A1 Fused pyramidine derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-11 US disclosed
US-20070010537-A1 Fused pyramidine derivative and use thereof TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2007-01-11 US disclosed
EP-1657238-A1 FUSED PYRIMIDINE DERIVATIVE AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2006-05-17 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070010537-A1 Fused pyramidine derivative and use thereof NR5A1, GNRHR, RXFP3 DDX3X 3247/4885CYP3A4 1715/4885CYP2C9 2416/4885
US-20180333376-A1 USE OF (BENZENESULFONAMIDO) BENZAMIDE COMPOUNDS FOR INHIBITING LIVER FIBROSIS COL1A1, COL2A1, COL14A1 DDX3X 1763/4885CYP3A4 1098/4885CYP2C9 773/4885
US-20190274979-A2 USE OF (BENZENESULFONAMIDO)BENZAMIDE COMPOUNDS FOR INHIBITING LIVER FIBROSIS COL1A1, COL2A1, COL14A1 DDX3X 1763/4885CYP3A4 1098/4885CYP2C9 773/4885
US-10933038-B2 Use of (benzenesulfonamido) benzamide compounds for inhibiting liver fibrosis COL1A1, COL2A1, COL14A1 DDX3X 1763/4885CYP3A4 1098/4885CYP2C9 773/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.