SCHEMBL5470632

SCHEMBL5470632

COc1ccccc1N1C(=O)CCN(Cc2ccc(N)cc2)C1=O

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.51
MAPK1 P28482 1/20 0.44
ADRA1D P25100 4/20 0.43
ADRA1A P35348 4/20 0.43
ADRA1B P35368 1/20 0.42
MAPT P10636 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
MGLL Q99685 1/20 0.42
MEN1 O00255 1/20 0.41
CYP1A2 P05177 1/20 0.41
HTR1A P08908 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
HTR7 P34969 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5484204 0.84 SMN1; SMN2 (0.48) POLBMAPK1ADRA1DADRA1AADRA1B
SCHEMBL5480222 0.84 POLB (0.57) POLBMAPK1ADRA1DADRA1AADRA1B
SCHEMBL5482189 0.82 POLB (0.47) POLBMAPK1SMN1; SMN2MEN1HTR7
SCHEMBL5477807 0.76 POLB (0.55) POLBMAPK1MEN1KMT2A
SCHEMBL5482627 0.72 POLB (0.53) POLBMAPTMEN1CYP2C9CYP2C19
SCHEMBL19561754 0.72 MAPK1 (0.80) MAPK1HTR7KMT2A
SCHEMBL8152227 0.72 ATM (0.52) POLBMAPTMGLLMEN1CYP1A2
SCHEMBL5474190 0.72 ENPP2 (0.51) POLBMAPTSMN1; SMN2MGLLMEN1
SCHEMBL11431546 0.72 MGLL (0.57) POLBMAPTSMN1; SMN2MGLLMEN1
SCHEMBL13533230 0.70 ADRA1D (0.77) MAPK1ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20070010529-A1 Nitrogenous heterocyclic compounds and medical use thereof ONO PHARMACEUTICAL CO., LTD. (JP) 2007-01-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070010529-A1 Nitrogenous heterocyclic compounds and medical use thereof MAPK1, NOS1, NOS2 POLB 2709/4885MAPK1 1/4885ADRA1D 2776/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.