SCHEMBL5505355

SCHEMBL5505355

CCCN1C(=O)C([Fe])c2cc(N)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 7/20 0.43
ALDH1A1 P00352 4/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41
ATAD2 Q6PL18 1/20 0.38
CHEK1 O14757 1/20 0.38
AURKA O14965 1/20 0.38
DAPK3 O43293 1/20 0.38
JAK2 O60674 1/20 0.38
PRKD3 O94806 1/20 0.38
MAP4K4 O95819 1/20 0.38
PAK4 O96013 1/20 0.38
ABL1 P00519 1/20 0.38
NTRK1 P04629 1/20 0.38
LCK P06239 1/20 0.38
FYN P06241 1/20 0.38
CSF1R P07333 1/20 0.38
RET P07949 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5506950 0.80 CHEK1 (0.50) CYP19A1ALDH1A1ATAD2CHEK1AURKA
SCHEMBL20548712 0.75 CYP19A1 (0.39) CYP19A1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5505345 0.74 CYP19A1 (0.36) CYP19A1CNR2CNR1
SCHEMBL20616486 0.74 CYP19A1 (0.38) CYP19A1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL20335475 0.74 CYP19A1 (0.50) CYP19A1ALDH1A1CYP1A2CYP3A4CYP2D6
SCHEMBL5503471 0.73 CHEK1 (0.36) ALDH1A1ATAD2CHEK1AURKADAPK3
SCHEMBL5501204 0.70 CHEK1 (0.33) ATAD2CHEK1AURKADAPK3JAK2
SCHEMBL28070866 0.69 ACVR1 (0.45) CYP19A1ALDH1A1CYP1A2ATAD2CHEK1
SCHEMBL3648722 0.68 PARK7 (0.50) ALDH1A1MAPTCA12CA1CA2
SCHEMBL5116351 0.67 ATAD2 (0.57) CYP19A1ALDH1A1ATAD2ACVR1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1781642-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS Pharmacia & Upjohn Company LLC (US) 2007-05-09 EP disclosed
WO-2006016221-A1 OXAZOLIDINONES CONTAINING OXINDOLES AS ANTIBACTERIAL AGENTS PHARMACIA & UPJOHN COMPANY LLC (US) 2006-02-16 WO disclosed