SCHEMBL5518599

SCHEMBL5518599

CC(C)C[C@H](OCc1ccccc1-c1ccc(-c2ccc(-n3ccnc3)cc2)cc1)C(=O)NCC#N

nearest known ligand 0.46

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
PORCN Q9H237 6/20 0.46
CTSK P43235 5/20 0.42
CTSS P25774 4/20 0.42
CTSB P07858 4/20 0.41
CTSL P07711 4/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
ADH5 P11766 3/20 0.40
MEN1 O00255 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
KMT2A Q03164 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6178943 0.82 CTSK (0.48) PORCNCTSKCTSSCTSBCTSL
SCHEMBL5516782 0.82 CTSK (0.48) PORCNCTSKCTSSCTSBCTSL
SCHEMBL6001121 0.81 CTSB (0.53) CTSKCTSSCTSBCTSL
SCHEMBL4700947 0.79 CTSL (0.66) CTSKCTSSCTSBCTSL
SCHEMBL6172215 0.79 CTSK (0.58) CTSKCTSSCTSBCTSL
SCHEMBL4700794 0.76 CTSS (0.62) CTSKCTSSCTSBCTSL
SCHEMBL5514860 0.75 CTSS (0.44) CTSKCTSSCTSBCTSL
SCHEMBL4700791 0.74 CTSS (0.45) CTSKCTSSCTSBCTSL
SCHEMBL4699259 0.73 CTSK (0.60) CTSKCTSSCTSBCTSL
SCHEMBL6208701 0.72 CTSS (0.48) CTSKCTSSCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7279478-B2 Cathepsin cysteine protease inhibitors MERCK FROSST CANADA & CO. (CA) 2007-10-09 US disclosed